SCHEMBL11538709

SCHEMBL11538709

Cc1cccc(Cl)c1-n1cnnc1S

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.38
CHRNA7 P36544 12/20 0.36
HSD11B1 P28845 1/20 0.35
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11537274 0.81 MEN1 (0.36) P2RX7HSD11B1LMNATSHRMAPK1
SCHEMBL14112935 0.73 PI4KA (0.40) ALDH1A1TSHR
SCHEMBL11537218 0.73 HCAR1 (0.40) P2RX7HSD11B1ALDH1A1
SCHEMBL1493493 0.71 ALDH1A1 (0.47) P2RX7ALDH1A1LMNAALOX15TSHR
SCHEMBL11091625 0.70 HCAR1 (0.40) ALDH1A1TSHR
SCHEMBL14204026 0.67 FGFR1 (0.47) ALDH1A1HTT
SCHEMBL11538267 0.66 NOTUM (0.38) HSD11B1ALDH1A1LMNATSHRHTT
SCHEMBL14951333 0.65 P2RX7 (0.36) P2RX7ALDH1A1LMNAALOX15TSHR
SCHEMBL14112937 0.65 MAPK1 (0.43) MAPK1
SCHEMBL2550381 0.65 NOTUM (0.46) ALDH1A1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4134914-A 1-Acyl-4-substituted phenyl thiosemicarbazides ELI LILLY AND COMPANY (US) 1979-01-16 US disclosed
US-4082762-A 4-(2-HALOPHENYL)-1,2,4-TRIAZOLE-3-THIOL COMPOUNDS ELI LILLY AND COMPANY (US) 1978-04-04 US disclosed
US-3937713-A Process for the preparation of s-triazolo[3,4-b]benzothiazoles ELI LILLY AND COMPANY (US) 1976-02-10 US disclosed