SCHEMBL11538804

SCHEMBL11538804

COc1ccc2cc(C(C)C(=O)c3ccccc3)ccc2c1

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.70
AKR1C3 P42330 6/20 0.70
AKR1C2 P52895 6/20 0.70
PTGS1 P23219 3/20 0.70
TSHR P16473 2/20 0.70
CDC42 P60953 1/20 0.70
RAC1 P63000 1/20 0.70
CYP1A2 P05177 1/20 0.70
SLC22A6 Q4U2R8 1/20 0.70
LMNA P02545 1/20 0.62
MAPT P10636 1/20 0.62
CYP2C9 P11712 1/20 0.62
TDP1 Q9NUW8 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
AKR1C1 Q04828 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30076171 0.86 UGT2B7 (0.55) PTGS2AKR1C3AKR1C2PTGS1TSHR
SCHEMBL4808086 0.86 UGT2B7 (0.55) PTGS2AKR1C3AKR1C2PTGS1TSHR
SCHEMBL1755267 0.86 L3MBTL1 (0.58) PTGS2AKR1C3AKR1C2PTGS1TSHR
SCHEMBL6510993 0.85 PTGS1 (0.56) PTGS2PTGS1MAPTMEN1KMT2A
Naproxen SCHEMBL23753934 0.84 AKR1C3 (0.88) PTGS2AKR1C3AKR1C2PTGS1TSHR
Naproxen SCHEMBL28881206 0.84 AKR1C3 (0.88) PTGS2AKR1C3AKR1C2PTGS1TSHR
SCHEMBL9246980 0.83 PTGS2 (0.63) PTGS2AKR1C3AKR1C2PTGS1TSHR
SCHEMBL12090351 0.83 PTGS2 (0.63) PTGS2AKR1C3AKR1C2PTGS1TSHR
Naproxen SCHEMBL616149 0.83 AKR1C3 (1.00) PTGS2AKR1C3AKR1C2PTGS1TSHR
Naproxen SCHEMBL3046 0.83 AKR1C3 (1.00) PTGS2AKR1C3AKR1C2PTGS1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4142054-A TRIVALENT THALLIUM SALT THE UPJOHN COMPANY (US) 1979-02-27 US disclosed
US-4135051-A ENOL ETHER OF AN ARYL ALKYL KETONE WITH A THALLIJM SALT, REGENERATION OF THALLIUM SALT BY ADDING PERACID AND REACTIVE METAL COMPOUND THE UPJOHN COMPANY (US) 1979-01-16 US disclosed
US-4107439-A Process for preparing arylalkanoic acid derivatives THE UPJOHN COMPANY (US) 1978-08-15 US disclosed