SCHEMBL11539823

SCHEMBL11539823

CC(=O)Oc1cc(=O)n(-c2ccc(C(F)(F)F)cc2)c2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.49
PPARG P37231 5/20 0.47
PPARA Q07869 3/20 0.47
HPGD P15428 3/20 0.43
HSD17B10 Q99714 2/20 0.43
USP2 O75604 2/20 0.43
ALDH1A1 P00352 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP2C19 P33261 1/20 0.43
BRD4 O60885 1/20 0.40
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HTT P42858 1/20 0.39
MAT2A P31153 1/20 0.38
TEAD1 P28347 1/20 0.38
TEAD4 Q15561 1/20 0.38
TEAD2 Q15562 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11543287 0.88 HPGD (0.50) BACE1PPARGPPARAHPGDHSD17B10
SCHEMBL11544309 0.87 BACE1 (0.48) BACE1PPARGPPARAHPGDHSD17B10
SCHEMBL11542615 0.86 NPSR1 (0.46) NPSR1BRD4MEN1KMT2AHTT
SCHEMBL11540274 0.86 NPSR1 (0.47) HPGDHSD17B10ALDH1A1NPSR1KDM4E
SCHEMBL11541055 0.84 NPSR1 (0.46) HPGDHSD17B10ALDH1A1NPSR1KDM4E
SCHEMBL11540070 0.84 NPSR1 (0.46) HPGDHSD17B10ALDH1A1NPSR1KDM4E
SCHEMBL11538165 0.83 NPSR1 (0.51) BACE1PPARGHPGDNPSR1KDM4E
SCHEMBL11541058 0.81 ALDH1A1 (0.42) BACE1HSD17B10ALDH1A1KDM4EBRD4
SCHEMBL25042634 0.78 KDM4E (0.50) PPARGPPARAHPGDALDH1A1KDM4E
SCHEMBL11544638 0.78 THRB (0.45) HPGDHSD17B10USP2ALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4168312-A Quinolone derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-09-18 US claimed
US-4168312-A Quinolone derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-09-18 US disclosed