SCHEMBL11540608

SCHEMBL11540608

O=C(O)c1cc2c(OCC(O)CN3CCC(COc4ccccc4)CC3)cccc2[nH]1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 8/20 0.55
ADRB1 P08588 7/20 0.55
ADRB3 P13945 7/20 0.55
DRD4 P21917 6/20 0.53
DRD2 P14416 5/20 0.53
ALDH1A1 P00352 1/20 0.52
MAPT P10636 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
DRD3 P35462 3/20 0.48
SRD5A2 P31213 1/20 0.48
HTR1A P08908 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11541108 0.90 ADRB2 (0.51) ADRB2ADRB1ADRB3DRD4DRD2
SCHEMBL11543042 0.87 HTR1A (0.62) ADRB2ADRB1ADRB3DRD4DRD2
Benzoic Acid SCHEMBL11538250 0.87 HTR1A (0.57) ADRB2ADRB1ADRB3DRD4DRD2
Benzoic Acid SCHEMBL11543852 0.87 ADRB2 (0.53) ADRB2ADRB1ADRB3DRD4DRD2
SCHEMBL11537345 0.86 DRD4 (0.56) ADRB2ADRB1ADRB3DRD4DRD2
SCHEMBL11543858 0.84 ADRB2 (0.53) ADRB2ADRB1ADRB3DRD4DRD2
SCHEMBL5584614 0.83 HTR1A (0.60) ADRB2ADRB1ADRB3DRD4DRD2
SCHEMBL5584230 0.83 HTR1A (0.60) ADRB2ADRB1ADRB3DRD4DRD2
SCHEMBL5584233 0.83 HTR1A (0.60) ADRB2ADRB1ADRB3DRD4DRD2
SCHEMBL11537853 0.83 ADRB2 (0.49) ADRB2ADRB1ADRB3DRD4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4146630-A HYPOTENSIVE AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1979-03-27 US disclosed