SCHEMBL11543045

SCHEMBL11543045

CNC(=O)N(S)c1cccc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.49
SIGMAR1 Q99720 5/20 0.46
GAA P10253 3/20 0.45
ALDH1A1 P00352 3/20 0.45
PGR P06401 1/20 0.45
PTGS1 P23219 1/20 0.45
MAPK1 P28482 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MTNR1A P48039 2/20 0.41
MMP9 P14780 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
KDM4E B2RXH2 2/20 0.39
MMP3 P08254 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
NR4A1 P22736 1/20 0.38
NR4A2 P43354 1/20 0.38
NR4A3 Q92570 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28851168 0.81 SIGMAR1 (0.61) PLK1SIGMAR1GAAALDH1A1PGR
SCHEMBL28068452 0.81 SIGMAR1 (0.50) PLK1SIGMAR1GAAALDH1A1MTNR1A
SCHEMBL11360909 0.78 SIGMAR1 (0.51) PLK1SIGMAR1GAANR4A1NR4A2
SCHEMBL10492074 0.78 SIGMAR1 (0.57) PLK1SIGMAR1GAAALDH1A1PGR
SCHEMBL11541431 0.77 TP53 (0.39) GAAALDH1A1SLC6A2SLC6A4KDM4E
SCHEMBL5966385 0.77 SIGMAR1 (0.46) SIGMAR1GAAALDH1A1MTNR1AMMP9
SCHEMBL11131086 0.76 SIGMAR1 (0.46) PLK1SIGMAR1GAAALDH1A1PGR
SCHEMBL11542282 0.76 ALDH1A1 (0.38) GAAALDH1A1HSD17B10SLC6A2SLC6A4
SCHEMBL11514484 0.75 LMNA (0.35) PLK1HDAC8
SCHEMBL11548288 0.75 ALDH1A1 (0.39) ALDH1A1PTGS1MAPK1HSD17B10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4148799-A Process for the preparation of 2-aryliminothiazoline solutions BAYER AKTIENGESELLSCHAFT (DE) 1979-04-10 US disclosed