SCHEMBL11544340

SCHEMBL11544340

O=C(OC(=O)[C@@H]1CCCN1)C(CS)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C19 P33261 1/20 0.44
SLC6A3 Q01959 8/20 0.42
SLC6A2 P23975 6/20 0.42
SLC6A4 P31645 4/20 0.42
ELANE P08246 1/20 0.41
TSHR P16473 2/20 0.41
CYP2C9 P11712 1/20 0.41
DHFR P00374 1/20 0.41
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CTSC P53634 1/20 0.40
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11546126 0.82 SLC6A3 (0.43) CYP3A4CYP2D6CYP1A2CYP2C19SLC6A3
SCHEMBL7381712 0.81 CTSC (0.48) ELANEALDH1A1CTSCHTR2CHTR2B
SCHEMBL11406016 0.79 CYP3A4 (0.46) CYP3A4CYP2D6CYP1A2CYP2C19SLC6A3
SCHEMBL11248554 0.78 CYP3A4 (0.44) CYP3A4CYP2D6CYP1A2CYP2C19SLC6A3
SCHEMBL11433291 0.77 CPN1 (0.38) ELANE
SCHEMBL7377900 0.76 CTSC (0.47) CYP3A4CYP2D6CYP1A2CYP2C19SLC6A3
SCHEMBL11558863 0.76 CTSC (0.51) CYP3A4CYP2D6CYP1A2CYP2C19SLC6A3
SCHEMBL11489216 0.76 ELANE (0.40) CYP3A4CYP2D6CYP1A2CYP2C19SLC6A3
SCHEMBL11430086 0.76 NOS2 (0.33) CYP3A4CYP2D6CYP1A2CYP2C19ELANE
SCHEMBL11438879 0.76 NOS2 (0.33) CYP3A4CYP2D6CYP1A2CYP2C19ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4154840-A Antihypertensive pipecolic acid derivatives E. R. SQUIBB & SONS, INC. (US) 1979-05-15 US disclosed
US-4105776-A ANGIOTENSIN CONVERTING ENZYME INHIBITORS, HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1978-08-08 US disclosed