SCHEMBL11544600

SCHEMBL11544600

O=C1OCCCC1N1C(=O)c2cccc3cccc(c23)C1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.51
ALDH1A1 P00352 7/20 0.51
ERCC1 P07992 1/20 0.42
FEN1 P39748 1/20 0.42
ERCC4 Q92889 1/20 0.42
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 3/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
HPGD P15428 4/20 0.40
CYP1A2 P05177 2/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
AKR1B1 P15121 1/20 0.40
ALOX15 P16050 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11538199 0.91 TSHR (0.49) KDM4EALDH1A1ERCC1FEN1ERCC4
SCHEMBL9624719 0.77 TSHR (0.59) ALDH1A1GAATSHRHSD17B10HPGD
SCHEMBL29386585 0.69 TYMS (0.59) KDM4EALDH1A1ERCC1FEN1ERCC4
SCHEMBL2175176 0.69 CRBN (0.78) ALDH1A1TSHRCYP1A2
SCHEMBL4256711 0.68 ALDH1A1 (1.00) KDM4EALDH1A1GAATSHRHSD17B10
SCHEMBL11542774 0.67 ERCC1 (0.51) KDM4EALDH1A1ERCC1FEN1ERCC4
SCHEMBL11537599 0.67 ERCC1 (0.51) KDM4EALDH1A1ERCC1FEN1ERCC4
SCHEMBL11537593 0.67 ERCC1 (0.51) KDM4EALDH1A1ERCC1FEN1ERCC4
SCHEMBL27538862 0.67 ALDH1A1 (0.46) KDM4EALDH1A1ERCC1FEN1ERCC4
SCHEMBL9876170 0.66 KDM4E (0.42) KDM4EALDH1A1ERCC1FEN1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4180579-A 2-Substituted-1H-benz[de]-isoquinoline-1,3(2H)-diones E. R. SQUIBB & SONS, INC. (US) 1979-12-25 US disclosed
US-4170651-A ANTIINFLAMMATORY AGENTS E. R. SQUIBB & SONS, INC. (US) 1979-10-09 US disclosed
US-4115555-A ANTIINFLAMMATORY E. R. SQUIBB & SONS, INC. (US) 1978-09-19 US disclosed
US-4051246-A ANTIINFLAMMATORY E. R. SQUIBB & SONS, INC. (US) 1977-09-27 US disclosed