SCHEMBL11544907

SCHEMBL11544907

O=C(c1ccccc1)c1cc2c3ccccc3[nH]c(=O)n2n1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 10/20 0.69
GRIN2D O15399 1/20 0.51
GRIN3B O60391 1/20 0.51
GRIA1 P42261 1/20 0.51
GRIA2 P42262 1/20 0.51
GRIA3 P42263 1/20 0.51
GRIA4 P48058 1/20 0.51
GRIN1 Q05586 1/20 0.51
GRIN2A Q12879 1/20 0.51
GRIN2B Q13224 1/20 0.51
GRIN2C Q14957 1/20 0.51
GRIN3A Q8TCU5 1/20 0.51
GABRP O00591 1/20 0.47
GABRD O14764 1/20 0.47
GABRA1 P14867 1/20 0.47
GABRB1 P18505 1/20 0.47
GABRG2 P18507 1/20 0.47
GABRB3 P28472 1/20 0.47
GABRA5 P31644 1/20 0.47
GABRA3 P34903 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11258739 0.88 ADORA3 (0.74) ADORA3GRIN2DGRIN3BGRIA1GRIA2
SCHEMBL11255156 0.84 ADORA3 (0.76) ADORA3GRIN2DGRIN3BGRIA1GRIA2
SCHEMBL11258237 0.84 ADORA3 (0.72) ADORA3GRIN2DGRIN3BGRIA1GRIA2
SCHEMBL11250907 0.84 ADORA3 (0.72) ADORA3GRIN2DGRIN3BGRIA1GRIA2
Acetone SCHEMBL11543246 0.83 ADORA3 (0.74) ADORA3GRIN2DGRIN3BGRIA1GRIA2
Acetaldehyde SCHEMBL11543250 0.80 ADORA3 (0.70) ADORA3GRIN2DGRIN3BGRIA1GRIA2
SCHEMBL11631304 0.78 ADORA3 (0.67) ADORA3
SCHEMBL11631308 0.78 ADORA3 (0.67) ADORA3
SCHEMBL11266931 0.78 ADORA3 (1.00) ADORA3GABRPGABRDGABRA1GABRB1
SCHEMBL11250103 0.76 ADORA3 (0.58) ADORA3GABRPGABRDGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4179561-A REACTING A 3-DIAZOOXINDOLE WITH A SUBSTITUTED ACETYLENE E. R. SQUIBB & SONS, INC. (US) 1979-12-18 US disclosed
US-4163789-A Anti-psychotic (cycloalkenylalkylpiperidino) benzamides ANPHAR, S.A. (ES) 1979-08-07 US disclosed
US-4112096-A ANTIALLERGENS E. R. SQUIBB & SONS, INC. (US) 1978-09-05 US disclosed
US-4076818-A ANTIALLERGENS E. R. SQUIBB & SONS, INC. (US) 1978-02-28 US disclosed