SCHEMBL11545209

SCHEMBL11545209

Cc1cccnc1OCC(O)CNCCOc1ccc(C(N)=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.53
ADRB1 P08588 8/20 0.50
ADRB3 P13945 5/20 0.50
ADRB2 P07550 5/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
ABCB1 P08183 2/20 0.44
HSD17B10 Q99714 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11547450 0.89 ATM (0.48) ATMADRB1ADRB3ADRB2CYP1A2
SCHEMBL11546061 0.88 ATM (0.53) ATMADRB1ADRB3ADRB2CYP1A2
SCHEMBL11549194 0.87 ATM (0.48) ATMADRB1ADRB3ADRB2CYP1A2
SCHEMBL11547629 0.86 ATM (0.53) ATMADRB1ADRB3ADRB2CYP1A2
SCHEMBL10714000 0.85 ADRB2 (0.58) ATMADRB1ADRB3ADRB2CYP1A2
SCHEMBL11547838 0.85 ADRB1 (0.56) ATMADRB1ADRB3ADRB2CYP1A2
SCHEMBL11550779 0.85 ADRB3 (0.54) ATMADRB1ADRB3ADRB2CYP1A2
SCHEMBL11548208 0.85 ATM (0.53) ATMADRB1ADRB3ADRB2CYP1A2
Tolamolol SCHEMBL611643 0.84 ATM (0.59) ATMADRB1ADRB3ADRB2CYP1A2
Tolamolol SCHEMBL613511 0.84 ATM (0.59) ATMADRB1ADRB3ADRB2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139623-A HYPOTENSIVE AGENTS C-G CORP. (US) 1979-02-13 US disclosed
US-4027027-A BETA-RECEPTOR-BLOCKERS, HYPOTENSIVES AND VALODILATORS; FOR TREATING ARRYTHMIAS AND ANGINA PECTORIS CIBA-GEIGY CORPORATION (US) 1977-05-31 US disclosed