SCHEMBL11546751

SCHEMBL11546751

CNS(=O)(=O)c1cc(C(=O)OC)cc(N)c1Oc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.49
HPGD P15428 5/20 0.49
KDM4E B2RXH2 4/20 0.49
GAA P10253 3/20 0.49
PKM P14618 1/20 0.49
USP2 O75604 3/20 0.43
ACLY P53396 5/20 0.41
HSD17B10 Q99714 4/20 0.40
LMNA P02545 3/20 0.40
TSHR P16473 2/20 0.40
HIF1A Q16665 2/20 0.40
CA2 P00918 1/20 0.40
BLM P54132 1/20 0.40
SLC12A2 P55011 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MAPT P10636 2/20 0.40
GLA P06280 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
ATM Q13315 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11849419 0.90 ALDH1A1 (0.49) ALDH1A1HPGDKDM4EGAAPKM
SCHEMBL2875469 0.88 HPGD (0.52) ALDH1A1HPGDKDM4EGAAPKM
SCHEMBL14879659 0.88 ALDH1A1 (0.51) ALDH1A1HPGDKDM4EGAAPKM
SCHEMBL573278 0.84 ALDH1A1 (0.48) ALDH1A1HPGDKDM4EGAAPKM
SCHEMBL11545452 0.84 USP2 (0.54) ALDH1A1HPGDKDM4EGAAPKM
SCHEMBL11546591 0.80 ALDH1A1 (0.62) ALDH1A1HPGDKDM4EGAAUSP2
SCHEMBL574175 0.79 HPGD (0.43) ALDH1A1HPGDKDM4EGAAPKM
SCHEMBL573731 0.79 HPGD (0.43) ALDH1A1HPGDKDM4EGAAPKM
SCHEMBL11550368 0.79 ALDH1A1 (0.43) ALDH1A1HPGDKDM4EUSP2ACLY
SCHEMBL11847444 0.78 ALDH1A1 (0.47) ALDH1A1HPGDKDM4EGAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4161531-A Diuretic and saluretic 5-sulfamoylbenzoic acid derivatives carrying a heterocyclic substituent HOECHST AKTIENGESELLSCHAFT (DE) 1979-07-17 US disclosed
US-4118397-A DIURETICS HOECHST AKTIENGESELLSCHAFT (DE) 1978-10-03 US disclosed
US-4111953-A DIURETICS HOECHST AKTIENGESELLSCHAFT (DE) 1978-09-05 US disclosed
US-4093735-A DIURETICS HOECHST AKTIENGESELLSCHAFT (DT) 1978-06-06 US disclosed
US-4010273-A DIURETICS, SALURETICS HOECHST AKTIENGESELLSCHAFT (DT) 1977-03-01 US disclosed