SCHEMBL11547645

SCHEMBL11547645

O=C(CCSCCc1ccccc1)OC(=O)[C@@H]1CCCN1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
CTSC P53634 1/20 0.41
ELANE P08246 1/20 0.40
GBA1 P04062 2/20 0.38
KDM4E B2RXH2 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
DPP4 P27487 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
CES1 P23141 1/20 0.35
MMP12 P39900 1/20 0.35
MMP13 P45452 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7582887 0.89 TDP1 (0.46) HTR2CHTR2BCTSCELANETSHR
SCHEMBL11549982 0.85 HTR2C (0.42) HTR2CHTR2BCTSCTSHRTAAR1
SCHEMBL7386495 0.84 CYP2C19 (0.42) HTR2CHTR2BCTSCELANEGBA1
SCHEMBL11545881 0.83 IDO1 (0.43) HTR2CHTR2BCTSCELANEKDM4E
SCHEMBL7379917 0.81 KMT2A (0.42) HTR2CHTR2BCTSCELANEKDM4E
SCHEMBL7373953 0.81 KMT2A (0.42) HTR2CHTR2BCTSCELANEKDM4E
SCHEMBL474619 0.81 HTR2C (0.47) HTR2CHTR2BCTSCELANETSHR
SCHEMBL11544707 0.80 SLC6A1 (0.41) HTR2CHTR2BCTSCELANEKDM4E
SCHEMBL28274418 0.80 HTR2C (0.46) HTR2CHTR2BCTSCELANETSHR
SCHEMBL11544261 0.79 ELANE (0.38) HTR2CHTR2BCTSCELANETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4154840-A Antihypertensive pipecolic acid derivatives E. R. SQUIBB & SONS, INC. (US) 1979-05-15 US disclosed
US-4105776-A ANGIOTENSIN CONVERTING ENZYME INHIBITORS, HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1978-08-08 US disclosed