SCHEMBL11544261

SCHEMBL11544261

O=C(CCSC(=O)Oc1ccccc1)OC(=O)[C@@H]1CCCN1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ELANE P08246 2/20 0.38
HTR2C P28335 3/20 0.38
DPP4 P27487 2/20 0.38
HTR2B P41595 2/20 0.38
DPP8 Q6V1X1 1/20 0.38
ANPEP P15144 1/20 0.38
CTSC P53634 1/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
GHSR Q92847 3/20 0.33
IDO1 P14902 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RAB9A P51151 1/20 0.33
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
SCN4A P35499 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7379917 0.84 KMT2A (0.42) ELANEHTR2CDPP4HTR2BDPP8
SCHEMBL7373953 0.84 KMT2A (0.42) ELANEHTR2CDPP4HTR2BDPP8
SCHEMBL11545881 0.81 IDO1 (0.43) ELANEHTR2CDPP4HTR2BDPP8
SCHEMBL11546196 0.81 ALDH1A1 (0.42) ELANEHTR2CDPP4HTR2BCTSC
SCHEMBL11546726 0.79 GHSR (0.38) ELANEHTR2CDPP4HTR2BDPP8
SCHEMBL11547645 0.79 HTR2C (0.42) ELANEHTR2CDPP4HTR2BDPP8
SCHEMBL11549982 0.78 HTR2C (0.42) HTR2CHTR2BCTSCALDH1A1RAB9A
SCHEMBL11544707 0.78 SLC6A1 (0.41) ELANEHTR2CDPP4HTR2BDPP8
SCHEMBL15155167 0.78 ELANE (0.46) ELANEHTR2CDPP4HTR2BDPP8
SCHEMBL7373153 0.77 KMT2A (0.39) ELANEHTR2CDPP4HTR2BDPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4154840-A Antihypertensive pipecolic acid derivatives E. R. SQUIBB & SONS, INC. (US) 1979-05-15 US disclosed
US-4105776-A ANGIOTENSIN CONVERTING ENZYME INHIBITORS, HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1978-08-08 US disclosed