SCHEMBL11544707

SCHEMBL11544707

O=C(CCSC(c1ccccc1)(c1ccccc1)c1ccccc1)OC(=O)[C@@H]1CCCN1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A1 P30531 1/20 0.41
SLC6A11 P48066 1/20 0.41
ELANE P08246 1/20 0.39
CYP2D6 P10635 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
HTR2C P28335 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
RAB9A P51151 1/20 0.36
HTR2B P41595 1/20 0.36
KIF11 P52732 9/20 0.36
CTSC P53634 1/20 0.35
CYP3A4 P08684 2/20 0.35
DPP4 P27487 2/20 0.34
DPP8 Q6V1X1 1/20 0.34
ANPEP P15144 1/20 0.34
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29503863 0.90 ELANE (0.38) SLC6A1SLC6A11ELANECYP2D6CYP1A2
SCHEMBL7379917 0.80 KMT2A (0.42) ELANECYP2D6CYP1A2CYP2C19HTR2C
SCHEMBL7373953 0.80 KMT2A (0.42) ELANECYP2D6CYP1A2CYP2C19HTR2C
SCHEMBL11547645 0.80 HTR2C (0.42) ELANECYP2D6CYP1A2CYP2C19HTR2C
SCHEMBL11546734 0.79 KIF11 (0.40) ELANECYP2D6CYP1A2CYP2C19KIF11
SCHEMBL11544261 0.78 ELANE (0.38) ELANECYP2D6CYP1A2CYP2C19HTR2C
SCHEMBL7582887 0.78 TDP1 (0.46) ELANECYP2D6CYP1A2CYP2C19HTR2C
SCHEMBL11546196 0.77 ALDH1A1 (0.42) ELANECYP2D6CYP1A2CYP2C19HTR2C
SCHEMBL11545881 0.77 IDO1 (0.43) ELANECYP2D6CYP1A2CYP2C19HTR2C
SCHEMBL11153901 0.77 KMT2A (0.47) ELANECYP2D6CYP1A2CYP2C19HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4154840-A Antihypertensive pipecolic acid derivatives E. R. SQUIBB & SONS, INC. (US) 1979-05-15 US disclosed
US-4105776-A ANGIOTENSIN CONVERTING ENZYME INHIBITORS, HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1978-08-08 US disclosed