SCHEMBL115477

SCHEMBL115477

Cc1cc(C)n(C(C=O)N2CCN(c3ccccc3-c3cnc(C)nc3)CC2)n1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 1/20 0.42
KCNH2 Q12809 1/20 0.42
DHFR P00374 3/20 0.34
HTR7 P34969 4/20 0.32
FEN1 P39748 1/20 0.32
MAPT P10636 1/20 0.32
USP2 O75604 1/20 0.31
TSHR P16473 1/20 0.31
HTR1A P08908 3/20 0.31
POLB P06746 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL115833 0.92 CXCR3 (0.41) CXCR3KCNH2DHFRFEN1POLB
SCHEMBL113252 0.91 CXCR3 (0.41) CXCR3KCNH2DHFRHTR7FEN1
SCHEMBL113125 0.90 CXCR3 (0.40) CXCR3KCNH2DHFRFEN1MAPT
SCHEMBL113986 0.90 CXCR3 (0.40) CXCR3KCNH2DHFRHTR7FEN1
SCHEMBL113545 0.90 CXCR3 (0.42) CXCR3KCNH2DHFRHTR7FEN1
SCHEMBL114268 0.90 CXCR3 (0.40) CXCR3KCNH2DHFRHTR7FEN1
SCHEMBL114405 0.89 CXCR3 (0.39) CXCR3KCNH2MAPTUSP2TSHR
SCHEMBL114041 0.89 CXCR3 (0.39) CXCR3KCNH2DHFRFEN1MAPT
SCHEMBL114135 0.89 CXCR3 (0.41) CXCR3KCNH2HTR7MAPTHTR1A
SCHEMBL112035 0.88 CNR2 (0.42) CXCR3KCNH2FEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-A1 CXCR3 RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-03-07 EP disclosed
WO-2010126811-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-11-04 WO disclosed