SCHEMBL115833

SCHEMBL115833

Cc1cc(C)n(C(C=O)N2CCN(c3ccccc3-c3cnc(N)nc3)CC2)n1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 1/20 0.41
KCNH2 Q12809 1/20 0.41
DHFR P00374 8/20 0.41
FEN1 P39748 9/20 0.38
ALOX5AP P20292 8/20 0.38
PIK3CD O00329 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL115477 0.92 CXCR3 (0.42) CXCR3KCNH2DHFRFEN1POLB
SCHEMBL113252 0.89 CXCR3 (0.41) CXCR3KCNH2DHFRFEN1PIK3CA
SCHEMBL113125 0.89 CXCR3 (0.40) CXCR3KCNH2DHFRFEN1ALOX5AP
SCHEMBL113986 0.89 CXCR3 (0.40) CXCR3KCNH2DHFRFEN1
SCHEMBL113545 0.89 CXCR3 (0.42) CXCR3KCNH2DHFRFEN1PIK3CA
SCHEMBL114268 0.89 CXCR3 (0.40) CXCR3KCNH2DHFRFEN1ALOX5AP
SCHEMBL114041 0.88 CXCR3 (0.39) CXCR3KCNH2DHFRFEN1
SCHEMBL114405 0.88 CXCR3 (0.39) CXCR3KCNH2
SCHEMBL114135 0.87 CXCR3 (0.41) CXCR3KCNH2POLB
SCHEMBL112035 0.86 CNR2 (0.42) CXCR3KCNH2FEN1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-A1 CXCR3 RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-03-07 EP disclosed
WO-2010126811-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-11-04 WO disclosed