SCHEMBL114268

SCHEMBL114268

COc1ncc(-c2ccccc2N2CCN(C(C=O)n3nc(C)cc3C)CC2)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 1/20 0.40
KCNH2 Q12809 1/20 0.40
DHFR P00374 2/20 0.36
HTR1A P08908 7/20 0.34
HTR7 P34969 7/20 0.34
TP53 P04637 2/20 0.33
MAPT P10636 1/20 0.33
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
TSHR P16473 2/20 0.32
HPGD P15428 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PIK3CA P42336 1/20 0.32
JAK2 O60674 1/20 0.31
PRMT5 O14744 1/20 0.31
WDR77 Q9BQA1 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL114135 0.91 CXCR3 (0.41) CXCR3KCNH2HTR1AHTR7MAPT
SCHEMBL115477 0.90 CXCR3 (0.42) CXCR3KCNH2DHFRHTR1AHTR7
SCHEMBL113540 0.90 CXCR3 (0.40) CXCR3KCNH2DHFRHTR1AHTR7
SCHEMBL115324 0.89 KCNH2 (0.41) CXCR3KCNH2HTR1AHTR7PIK3CA
SCHEMBL114572 0.89 DHFR (0.33) CXCR3DHFRHTR1AHTR7TSHR
SCHEMBL115833 0.89 CXCR3 (0.41) CXCR3KCNH2DHFRALOX5APFEN1
SCHEMBL113245 0.88 AGER (0.36) CXCR3KCNH2DHFRHTR1AHTR7
SCHEMBL113054 0.88 TNIK (0.34) KCNH2DHFRTP53MAPTHPGD
SCHEMBL114734 0.88 MAPT (0.39) CXCR3KCNH2DHFRHTR1AHTR7
SCHEMBL113252 0.88 CXCR3 (0.41) CXCR3KCNH2DHFRHTR7MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-A1 CXCR3 RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-03-07 EP disclosed
WO-2010126811-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-11-04 WO disclosed