SCHEMBL11547765

SCHEMBL11547765

COc1cc(N)c(N)cc1C(=O)NC1CCN(CC2=CCC=CC2)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.58
CYP3A4 P08684 2/20 0.58
CYP1A2 P05177 1/20 0.58
ADRA2A P08913 1/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C9 P11712 1/20 0.58
DRD2 P14416 1/20 0.58
ADRA2B P18089 1/20 0.58
ADRA2C P18825 1/20 0.58
ACHE P22303 1/20 0.58
SLC6A2 P23975 1/20 0.58
HTR2A P28223 1/20 0.58
HTR2C P28335 1/20 0.58
ADRA1A P35348 1/20 0.58
DRD3 P35462 1/20 0.58
OPRK1 P41145 1/20 0.58
HTR2B P41595 1/20 0.58
CHRNA4 P43681 1/20 0.58
HTR3A P46098 1/20 0.58
SLC6A3 Q01959 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11551725 0.98 DRD4 (0.56) DRD4CYP3A4CYP1A2ADRA2ACYP2D6
SCHEMBL11543452 0.93 HTR4 (0.69) DRD4CYP3A4CYP1A2ADRA2ACYP2D6
SCHEMBL11550058 0.93 CYP3A4 (0.54) DRD4CYP3A4CYP1A2ADRA2ACYP2D6
Hydrochloric Acid SCHEMBL11548712 0.92 CYP3A4 (0.54) DRD4CYP3A4CYP1A2ADRA2ACYP2D6
Hydrochloric Acid SCHEMBL11545633 0.91 HTR4 (0.67) DRD4CYP3A4CYP1A2ADRA2ACYP2D6
SCHEMBL9865649 0.89 DRD2 (0.57) DRD4CYP3A4CYP1A2ADRA2ACYP2D6
Hydrochloric Acid SCHEMBL9866290 0.89 DRD2 (0.56) DRD4CYP3A4CYP1A2ADRA2ACYP2D6
SCHEMBL11552522 0.85 DRD2 (0.52) DRD4CYP3A4CYP1A2ADRA2ACYP2D6
SCHEMBL11545625 0.84 L3MBTL1 (0.47) DRD4CYP3A4CYP1A2ADRA2ACYP2D6
SCHEMBL11544379 0.84 DRD2 (0.54) DRD4CYP3A4CYP1A2ADRA2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4163789-A Anti-psychotic (cycloalkenylalkylpiperidino) benzamides ANPHAR, S.A. (ES) 1979-08-07 US claimed