SCHEMBL11547799

SCHEMBL11547799

COc1cc(NCCCC(C)N2C(=O)c3ccccc3C2=O)c2nc(C)cc(C)c2c1OC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.37
RAD52 P43351 1/20 0.36
MAPT P10636 2/20 0.35
GSK3B P49841 1/20 0.35
ESR1 P03372 1/20 0.34
PGR P06401 1/20 0.34
HTR1A P08908 1/20 0.34
DRD1 P21728 1/20 0.34
PTGS1 P23219 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
OPRM1 P35372 1/20 0.34
DRD3 P35462 1/20 0.34
SLC6A3 Q01959 1/20 0.34
TNF P01375 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HSP90AA1 P07900 2/20 0.34
HSP90AB1 P08238 2/20 0.34
MAOA P21397 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4728398 0.80 MEN1 (0.47) POLBRAD52MAPTGSK3BESR1
SCHEMBL6157510 0.79 ESR1 (0.63) MAPTGSK3BESR1PGRHTR1A
SCHEMBL11550294 0.79 MEN1 (0.48) POLBRAD52MAPTMEN1KMT2A
Hydrochloric Acid SCHEMBL11547653 0.78 HSP90AA1 (0.49) POLBRAD52MAPTMEN1KMT2A
Phosphoric Acid SCHEMBL11545454 0.77 RAD52 (0.50) POLBRAD52MAPTGSK3BESR1
SCHEMBL5496134 0.76 MAOA (0.60) RAD52GSK3BMEN1KMT2AHSP90AA1
SCHEMBL11543929 0.73 NSD2 (0.62) POLBRAD52MAPTHTR1AMEN1
Hydrochloric Acid SCHEMBL11544270 0.72 HSP90AA1 (0.67) POLBRAD52MAPTESR1PGR
SCHEMBL8660088 0.72 ESR1 (0.55) POLBMAPTGSK3BESR1PGR
SCHEMBL11544850 0.64 MAOA (0.47) GSK3BMAOAMAOBL3MBTL1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4167638-A Process for production of 8-NHR quinolines THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 1979-09-11 US disclosed