SCHEMBL6157510

SCHEMBL6157510

COc1cc(C)c2c(Oc3cccc(C(F)(F)F)c3)c(OC)cc(NCCCC(C)N3C(=O)c4ccccc4C3=O)c2n1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.63
PGR P06401 1/20 0.63
HTR1A P08908 1/20 0.63
DRD1 P21728 1/20 0.63
PTGS1 P23219 1/20 0.63
SLC6A2 P23975 1/20 0.63
SLC6A4 P31645 1/20 0.63
OPRM1 P35372 1/20 0.63
DRD3 P35462 1/20 0.63
SLC6A3 Q01959 1/20 0.63
GSK3B P49841 1/20 0.55
PRKD3 O94806 2/20 0.47
PRKCG P05129 2/20 0.47
PRKCB P05771 2/20 0.47
PRKCA P17252 2/20 0.47
PRKCH P24723 2/20 0.47
PRKCI P41743 2/20 0.47
PRKCE Q02156 2/20 0.47
PRKCQ Q04759 2/20 0.47
PRKCZ Q05513 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8660088 0.92 ESR1 (0.55) ESR1PGRHTR1ADRD1PTGS1
SCHEMBL5315847 0.86 ESR1 (0.72) ESR1PGRHTR1ADRD1PTGS1
SCHEMBL6156991 0.85 ESR1 (0.65) ESR1PGRHTR1ADRD1PTGS1
SCHEMBL5705813 0.84 ESR1 (0.75) ESR1PGRHTR1ADRD1PTGS1
SCHEMBL14424698 0.81 ESR1 (0.83) ESR1PGRHTR1ADRD1PTGS1
SCHEMBL11547799 0.79 POLB (0.37) ESR1PGRHTR1ADRD1PTGS1
SCHEMBL8656637 0.79 ESR1 (0.61) ESR1PGRHTR1ADRD1PTGS1
SCHEMBL19728197 0.78 ESR1 (0.86) ESR1PGRHTR1ADRD1PTGS1
SCHEMBL4354615 0.78 GSK3B (0.73) ESR1PGRHTR1ADRD1PTGS1
Tafenoquine SCHEMBL31160547 0.77 ESR1 (1.00) ESR1PGRHTR1ADRD1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501802-A2 PROCESS FOR THE PREPARATION OF QUINOLINE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 2005-02-02 EP disclosed
WO-2003093239-A2 PROCESS FOR THE PREPARATION OF QUINOLINE DERIVATIVES SMITHKLINE BEECHAM P.L.C. (GB) 2003-11-13 WO disclosed