SCHEMBL5496134

SCHEMBL5496134

COc1cc(NCCCC(C)N2C(=O)c3ccccc3C2=O)c2nccc(C)c2c1Oc1ccc(Cl)c(Cl)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 14/20 0.60
MAOB P27338 14/20 0.60
GSK3B P49841 1/20 0.50
PRKD3 O94806 1/20 0.42
PRKCG P05129 1/20 0.42
PRKCB P05771 1/20 0.42
PRKCA P17252 1/20 0.42
PRKCH P24723 1/20 0.42
PRKCI P41743 1/20 0.42
PRKCE Q02156 1/20 0.42
PRKCQ Q04759 1/20 0.42
PRKCZ Q05513 1/20 0.42
PRKCD Q05655 1/20 0.42
PRKD1 Q15139 1/20 0.42
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
NSD2 O96028 2/20 0.36
CASP6 P55212 2/20 0.36
RAD52 P43351 1/20 0.36
CASP7 P55210 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5496132 0.87 MAOA (0.54) MAOAMAOBGSK3BPRKD3PRKCG
SCHEMBL3856314 0.85 MAOA (0.70) MAOAMAOBGSK3BPRKD3PRKCG
SCHEMBL5493085 0.83 MAOA (0.72) MAOAMAOBGSK3BPRKD3PRKCG
SCHEMBL11543929 0.77 NSD2 (0.62) HSP90AA1HSP90AB1NSD2CASP6RAD52
SCHEMBL11547799 0.76 POLB (0.37) MAOAMAOBGSK3BHSP90AA1HSP90AB1
SCHEMBL14534511 0.75 MAOA (0.78) MAOAMAOBGSK3BPRKD3PRKCG
SCHEMBL6157510 0.75 ESR1 (0.63) MAOAMAOBGSK3BPRKD3PRKCG
SCHEMBL3856309 0.75 MAOA (1.00) MAOAMAOBGSK3BNSD2
SCHEMBL14443960 0.75 MAOA (1.00) MAOAMAOBGSK3BNSD2
SCHEMBL14443958 0.75 MAOA (1.00) MAOAMAOBGSK3BNSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0907363-B1 Medicament comprising (-)-8-[(4-amino-1-méthylbutyl)amino]-5-(3,4-dichlorophénoxy)-6-méthoxy-4-méthylquinoline for the treatment of parasitic and opportunistic infections UNIV MISSISSIPPI (US) 2007-05-23 EP disclosed
EP-0907363-A4 8-AMINOQUINOLINES UNIV MISSISSIPPI (US) 2005-04-06 EP disclosed
EP-0907363-A1 8-AMINOQUINOLINES THE UNIVERSITY OF MISSISSIPPI (US) 1999-04-14 EP disclosed
WO-1997036590-A1 8-AMINOQUINOLINES THE UNIVERSITY OF MISSISSIPPI (US) 1997-10-09 WO disclosed