SCHEMBL11549162

SCHEMBL11549162

Cc1ccccc1OCC(O)CNC(C)(C)COc1ccc(C(N)=O)cn1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 4/20 0.54
ADRB2 P07550 3/20 0.54
ADRB3 P13945 16/20 0.53
GRK3 P35626 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11545627 0.84 KDM4E (0.53) ADRB1ADRB2ADRB3GRK3
SCHEMBL11549323 0.83 KDM4E (0.49) ADRB1ADRB2ADRB3GRK3
SCHEMBL10892720 0.79 GRK3 (0.49) ADRB1ADRB2ADRB3GRK3
Hydrochloric Acid SCHEMBL10888073 0.78 GRK3 (0.49) ADRB1ADRB2ADRB3GRK3
SCHEMBL11545404 0.78 ADRB3 (0.41) ADRB1ADRB2ADRB3
SCHEMBL10889364 0.78 GRK3 (0.50) ADRB1ADRB2ADRB3GRK3
SCHEMBL11549703 0.75 ADRB2 (0.55) ADRB1ADRB2ADRB3GRK3
SCHEMBL10810577 0.75 ADRB2 (0.60) ADRB1ADRB2ADRB3
SCHEMBL11548953 0.75 OPRM1 (0.58)
SCHEMBL11550951 0.74 KDM4E (0.52) ADRB1ADRB2ADRB3GRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4027027-A BETA-RECEPTOR-BLOCKERS, HYPOTENSIVES AND VALODILATORS; FOR TREATING ARRYTHMIAS AND ANGINA PECTORIS CIBA-GEIGY CORPORATION (US) 1977-05-31 US claimed
US-4139623-A HYPOTENSIVE AGENTS C-G CORP. (US) 1979-02-13 US disclosed
US-4027027-A BETA-RECEPTOR-BLOCKERS, HYPOTENSIVES AND VALODILATORS; FOR TREATING ARRYTHMIAS AND ANGINA PECTORIS CIBA-GEIGY CORPORATION (US) 1977-05-31 US disclosed