SCHEMBL11554362

SCHEMBL11554362

CC(=O)Nc1cccnc1OCCNCC(O)COc1ccccc1C

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 2/20 0.49
ADRB1 P08588 3/20 0.46
ADRB3 P13945 3/20 0.46
ADRB2 P07550 2/20 0.46
GRK3 P35626 1/20 0.45
ATM Q13315 1/20 0.44
ABCB1 P08183 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11544327 0.85 KDM4E (0.52) KDM4EALDH1A1ADRB1ADRB3ADRB2
SCHEMBL11544470 0.83 ADRB2 (0.50) KDM4EALDH1A1ADRB1ADRB3ADRB2
SCHEMBL11547544 0.81 ADRB2 (0.53) KDM4EALDH1A1ADRB1ADRB3ADRB2
SCHEMBL11548885 0.80 KDM4E (0.47) KDM4EALDH1A1ADRB1ADRB3ADRB2
SCHEMBL11546543 0.80 ADRB2 (0.56) KDM4EALDH1A1ADRB1ADRB3ADRB2
SCHEMBL11548585 0.80 KDM4E (0.56) KDM4EALDH1A1ADRB1ADRB3ADRB2
Oxalic Acid SCHEMBL11546058 0.79 ALDH1A1 (0.64) KDM4EALDH1A1ADRB1ADRB3ADRB2
SCHEMBL11550521 0.79 KDM4E (0.47) KDM4EALDH1A1ADRB1ADRB3ADRB2
SCHEMBL11550779 0.79 ADRB3 (0.54) ALDH1A1ADRB1ADRB3ADRB2ATM
SCHEMBL11549370 0.77 ABCB1 (0.46) KDM4EALDH1A1ADRB1ADRB3ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139623-A HYPOTENSIVE AGENTS C-G CORP. (US) 1979-02-13 US disclosed
US-4027027-A BETA-RECEPTOR-BLOCKERS, HYPOTENSIVES AND VALODILATORS; FOR TREATING ARRYTHMIAS AND ANGINA PECTORIS CIBA-GEIGY CORPORATION (US) 1977-05-31 US disclosed