SCHEMBL11560283

SCHEMBL11560283

CC(C)c1[nH]c(=O)c(C#N)c2c1C(=O)c1ccccc1-2

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 5/20 0.41
PDE1C Q14123 1/20 0.41
ALDH1A1 P00352 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
KDM4E B2RXH2 5/20 0.39
ATM Q13315 2/20 0.39
GAA P10253 3/20 0.39
GLA P06280 2/20 0.39
IDO1 P14902 1/20 0.39
USP8 P40818 1/20 0.38
USP7 Q93009 1/20 0.38
PIM1 P11309 3/20 0.38
POLB P06746 1/20 0.38
BIRC5 O15392 1/20 0.37
HSD11B1 P28845 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11564817 0.82 PDE9A (0.46) PDE9APDE1CALDH1A1CYP1A2CYP2C9
SCHEMBL11568936 0.78 PDE9A (0.46) PDE9APDE1CALDH1A1CYP1A2CYP2C9
SCHEMBL11564514 0.77 HSD11B1 (0.56) PDE9AALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL11560285 0.76 ALDH1A1 (0.47) PDE9APDE1CALDH1A1CYP1A2CYP2C9
SCHEMBL11586131 0.74 KEAP1 (0.41) PDE9APDE1CALDH1A1CYP1A2CYP2C9
SCHEMBL11585656 0.72 KEAP1 (0.42) ALDH1A1HTTKDM4EATMIDO1
SCHEMBL11564415 0.72 USP8 (0.42) PDE9AALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL4277182 0.71 PDE9A (0.51) PDE9APDE1CALDH1A1CYP1A2CYP2C9
SCHEMBL5186477 0.70 PDE9A (0.47) PDE9APDE1CALDH1A1HTTKDM4E
SCHEMBL295307 0.69 ALDH1A1 (0.49) ALDH1A1CYP1A2CYP2C9CYP2C19HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4180666-A 3,9-Dihydro-3,9-dioxo-2H-indeno(2,1-c)-pyridine-4-(carbonitriles/carboxamides) G. D. SEARLE & CO. (US) 1979-12-25 US disclosed