SCHEMBL11564798

SCHEMBL11564798

O=[N+]([O-])c1nc(CC(O)CN2CCC(O)C2)c[nH]1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 3/20 0.35
CYP2D6 P10635 1/20 0.35
KDM4E B2RXH2 4/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
KCNA3 P22001 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17770528 0.85 L3MBTL1 (0.40) KDM4EALDH1A1LMNAMEN1KMT2A
SCHEMBL3814861 0.82 KMT2A (0.40) CYP2D6KDM4EALDH1A1POLBMEN1
SCHEMBL3811168 0.72 ALDH1A1 (0.39) ALDH1A1
SCHEMBL4635643 0.72 ALDH1A1 (0.31) ALDH1A1
SCHEMBL5682636 0.70 ALDH1A1 (0.44) KDM4EALDH1A1LMNAPOLBMEN1
SCHEMBL5681436 0.70 ALDH1A1 (0.44) KDM4EALDH1A1LMNAPOLBMEN1
SCHEMBL5681615 0.70 ALDH1A1 (0.44) KDM4EALDH1A1LMNAPOLBMEN1
SCHEMBL11350118 0.69 KMT2A (0.60) OPRK1CYP2D6KDM4ELMNAMEN1
SCHEMBL11569408 0.68 CA1 (0.30)
SCHEMBL6131556 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0000928-A1 Nitroimidazoles and pharmaceutical compositions containing them as well as their preparation F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1979-03-07 EP claimed
EP-0000928-A1 Nitroimidazoles and pharmaceutical compositions containing them as well as their preparation F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1979-03-07 EP disclosed