SCHEMBL11565358

SCHEMBL11565358

CCC(=O)N(c1ccc(C)cc1)C1(C(=O)OC)CCN(CCc2ccccc2)CC1

nearest known ligand 0.88

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 14/20 0.88
OPRD1 P41143 5/20 0.88
OPRK1 P41145 3/20 0.88
CACNA1C Q13936 1/20 0.68
OPRL1 P41146 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11565447 0.95 OPRM1 (0.86) OPRM1OPRD1OPRK1CACNA1COPRL1
Carfentanil SCHEMBL116222 0.94 OPRM1 (1.00) OPRM1OPRD1OPRK1CACNA1COPRL1
[11C]-Carfentanil SCHEMBL29374424 0.94 OPRM1 (1.00) OPRM1OPRD1OPRK1CACNA1COPRL1
SCHEMBL11563515 0.93 OPRM1 (0.78) OPRM1OPRD1OPRK1CACNA1C
Carfentanil SCHEMBL238456 0.93 OPRM1 (0.98) OPRM1OPRD1OPRK1CACNA1COPRL1
Carfentanil SCHEMBL4256090 0.93 OPRM1 (0.98) OPRM1OPRD1OPRK1CACNA1COPRL1
Carfentanil SCHEMBL9737212 0.92 OPRM1 (0.96) OPRM1OPRD1OPRK1CACNA1COPRL1
SCHEMBL11564695 0.91 OPRM1 (0.86) OPRM1OPRD1OPRK1CACNA1COPRL1
SCHEMBL11565029 0.91 OPRM1 (0.86) OPRM1OPRD1OPRK1CACNA1COPRL1
SCHEMBL11565614 0.89 OPRM1 (0.83) OPRM1OPRD1OPRK1CACNA1COPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4179569-A ANALGESIC INTERMEDIATES JANSSEN PHARMACEUTICA N.V. (BE) 1979-12-18 US disclosed
US-3998834-A ANALGESICS JANSSEN PHARMACEUTICA N.V. (BE) 1976-12-21 US disclosed