SCHEMBL11575869

SCHEMBL11575869

O=S(=O)(c1ccccc1)c1ccc2[nH]ncc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK3 O43781 1/20 0.54
CLK1 P49759 1/20 0.54
CLK2 P49760 1/20 0.54
CLK3 P49761 1/20 0.54
GSK3B P49841 1/20 0.54
CDK5 Q00535 1/20 0.54
DYRK1A Q13627 1/20 0.54
CDK5R1 Q15078 1/20 0.54
DYRK2 Q92630 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
DYRK1B Q9Y463 1/20 0.54
ROCK2 O75116 2/20 0.51
ROCK1 Q13464 2/20 0.51
RAB9A P51151 2/20 0.50
ALDH1A1 P00352 2/20 0.50
NPC1 O15118 1/20 0.50
JAK2 O60674 1/20 0.50
ACLY P53396 1/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15866404 0.81 NAMPT (0.47) DYRK3CLK2DYRK1ACLK4ROCK2
SCHEMBL30374957 0.80 ALDH1A1 (0.54) ALDH1A1NAMPTMAPTPOLBCDK2
SCHEMBL25179894 0.80 ALDH1A1 (0.54) ALDH1A1NAMPTMAPTPOLBCDK2
SCHEMBL1460717 0.79 ALDH1A1 (0.80) ROCK2ROCK1RAB9AALDH1A1NPC1
SCHEMBL3058692 0.78 MAPK1 (0.55) DYRK3CLK1CLK2CLK3GSK3B
SCHEMBL29509879 0.78 NOS1 (0.55) DYRK3CLK1CLK2CLK3GSK3B
SCHEMBL6298004 0.78 NOS1 (0.51) DYRK3CLK1CLK2CLK3GSK3B
SCHEMBL5220947 0.78 KDR (0.57) DYRK3CLK1CLK2CLK3GSK3B
SCHEMBL10179696 0.78 TMEM97 (0.52) DYRK3CLK1CLK2CLK3GSK3B
SCHEMBL31647068 0.78 KDR (0.57) DYRK3CLK1CLK2CLK3GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4096333-A NITROSATION OF A 2-METHYLACETANILIDE TENNECO CHEMICALS, INC. (US) 1978-06-20 US disclosed
US-3988347-A NITROSATION OF A 2-METHYL-ACETANILIDE WITH SODIUM NITRITE TENNECO CHEMICALS, INC. (US) 1976-10-26 US disclosed