SCHEMBL11577306

SCHEMBL11577306

CS(=O)(=O)CCN1C(=O)CN=C(c2ccccc2)c2cc(Cl)ccc21

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 4/20 0.67
KCNH2 Q12809 2/20 0.67
GABRP O00591 1/20 0.67
GABRD O14764 1/20 0.67
CACNA1F O60840 1/20 0.67
ALB P02768 1/20 0.67
GABRA1 P14867 1/20 0.67
GABRB1 P18505 1/20 0.67
GABRG2 P18507 1/20 0.67
GABRB3 P28472 1/20 0.67
GABRA5 P31644 1/20 0.67
GABRA3 P34903 1/20 0.67
AKR1C3 P42330 1/20 0.67
GABRA2 P47869 1/20 0.67
GABRB2 P47870 1/20 0.67
GABRA4 P48169 1/20 0.67
AKR1C2 P52895 1/20 0.67
GABRE P78334 1/20 0.67
CACNA1D Q01668 1/20 0.67
AKR1C1 Q04828 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11578526 0.94 OPRK1 (0.64) OPRK1KCNH2GABRPGABRDCACNA1F
SCHEMBL11577203 0.91 OPRK1 (0.65) OPRK1KCNH2GABRPGABRDCACNA1F
SCHEMBL11576383 0.89 OPRK1 (0.68) OPRK1KCNH2GABRPGABRDCACNA1F
SCHEMBL11576874 0.89 OPRK1 (0.63) OPRK1KCNH2GABRPGABRDCACNA1F
SCHEMBL11577976 0.88 TP53 (0.65) OPRK1KCNH2GABRPGABRDCACNA1F
SCHEMBL11578684 0.88 TP53 (0.57) OPRK1KCNH2GABRPGABRDCACNA1F
SCHEMBL11579241 0.87 GABRA1 (0.67) OPRK1KCNH2GABRPGABRDCACNA1F
SCHEMBL5361417 0.87 OPRK1 (0.72) OPRK1KCNH2GABRPGABRDCACNA1F
SCHEMBL11579759 0.87 OPRK1 (0.72) OPRK1KCNH2GABRPGABRDCACNA1F
SCHEMBL11578960 0.87 OPRK1 (0.63) OPRK1KCNH2GABRPGABRDCACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4010154-A Benzodiazepinones SUMITOMO CHEMICAL COMPANY, LIMITED (JA) 1977-03-01 US claimed
US-4079053-A Benzodiazepine derivatives SUMITOMO CHEMICAL COMPANY, LIMITED (JA) 1978-03-14 US disclosed
US-4010154-A Benzodiazepinones SUMITOMO CHEMICAL COMPANY, LIMITED (JA) 1977-03-01 US disclosed
US-3932637-A 1-ALKYLSULFONYLALKYL-1,4-BENZODIAZEPINONES SUMITOMO CHEMICAL COMPANY, LIMITED (JA) 1976-01-13 US disclosed