SCHEMBL11577633

SCHEMBL11577633

CSc1ccc2c(c1)C(=O)Cc1ccc(C)cc1O2

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.37
PTGS2 P35354 2/20 0.37
KDM4E B2RXH2 5/20 0.35
ATM Q13315 3/20 0.35
HTT P42858 2/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
METAP1 P53582 2/20 0.34
RAD52 P43351 1/20 0.33
TYMS P04818 1/20 0.33
MAOB P27338 6/20 0.33
HTR7 P34969 1/20 0.33
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11578024 0.90 KDM4E (0.36) PTGS1PTGS2KDM4EATMHTT
SCHEMBL9740773 0.83 MAOA (0.44) PTGS1PTGS2KDM4EATMHTT
SCHEMBL11576098 0.76 KDM4E (0.45) KDM4EATMHTTKMT2AMEN1
SCHEMBL11577085 0.76 MAOB (0.44) KDM4EKMT2AMEN1ALDH1A1HPGD
SCHEMBL11756804 0.73 ALDH1A1 (0.53) PTGS1PTGS2KDM4EATMHTT
SCHEMBL11124199 0.73 ALDH1A1 (0.41) KDM4EATMHTTKMT2AMEN1
SCHEMBL6906979 0.72 MAOA (0.46) KDM4EKMT2AMEN1ALDH1A1METAP1
SCHEMBL11759989 0.71 MEN1 (0.51) PTGS1PTGS2KDM4EATMHTT
SCHEMBL822842 0.71 METAP1 (0.44) PTGS1PTGS2HTTMETAP1TYMS
SCHEMBL11577980 0.70 MAOB (0.40) KDM4EATMHTTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4118572-A CNS DEPRESSANTS, NEUROLEPTIC AGENTS, SCHIZOPHRENIA, TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1978-10-03 US disclosed
US-4105664-A Dibenz[b,f]oxepin derivatives HOFFMANN-LA ROCHE INC. (US) 1978-08-08 US disclosed
US-4100173-A DEPRESSANTS, SCHIZOPHRENIA, TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1978-07-11 US disclosed
US-4091023-A ANTISCHIZOPHRENIA AGENTS, TRANQUILIZERS HOFFMANN-LA ROCHE INC. (US) 1978-05-23 US disclosed
US-4032525-A CNS DEPRESSANTS, NEUROLEPTICS HOFFMANN-LA ROCHE INC. (US) 1977-06-28 US disclosed