SCHEMBL11587730

SCHEMBL11587730

CCc1ccc2c(c1)C(CNC(=O)OC)c1cc(CC)ccc1C(F)(F)C2(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
TSHR P16473 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
SMN1; SMN2 Q16637 4/20 0.33
DRD2 P14416 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
HTR2C P28335 1/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11586182 0.80 EGFR (0.36) ALDH1A1TSHRTDP1SMN1; SMN2KDM4E
SCHEMBL11587643 0.78 PSEN1 (0.38) ALDH1A1TSHRSMN1; SMN2KDM4ELMNA
SCHEMBL11587446 0.78 PDK2 (0.40) KDM4EHTR2CMTNR1AMTNR1BLMNA
SCHEMBL11585655 0.77 AKR1C3 (0.36) ALDH1A1TSHRKDM4EGAAHTT
SCHEMBL11588154 0.76 APOB (0.37) ALDH1A1TSHRSMN1; SMN2KDM4ELMNA
SCHEMBL11587639 0.76 HPGD (0.35) ALDH1A1SMN1; SMN2KDM4ELMNAKMT2A
SCHEMBL11587156 0.73 HTR2A (0.39) DRD2HTR2CDRD1
SCHEMBL11588162 0.73 PDK2 (0.40) ALDH1A1SMN1; SMN2DRD2KDM4EGAA
SCHEMBL11586311 0.72 MC4R (0.34) ALDH1A1SMN1; SMN2KDM4EGAAHTT
SCHEMBL11587167 0.70 L3MBTL1 (0.37) TSHRTDP1SMN1; SMN2GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4070387-A ANTIARRHYTHMIC AGENTS MERCK & CO., INC. (US) 1978-01-24 US disclosed
US-4020096-A ANTIARRYTHMIA MERCK & CO., INC. (US) 1977-04-26 US disclosed
US-3950423-A 10,11-Dihydro-10,10,11,11-tetrafluoro-5H-dibenzo[a,d]cycloheptene-5-methylamines MERCK & CO., INC. (US) 1976-04-13 US disclosed