SCHEMBL11592378

SCHEMBL11592378

COc1cc(=O)[nH]c2nc(N)ccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.53
ADORA2A P29274 2/20 0.53
CA5A P35218 1/20 0.41
NQO2 P16083 3/20 0.40
CYP19A1 P11511 2/20 0.40
XDH P47989 1/20 0.39
MCHR1 Q99705 1/20 0.38
AR P10275 1/20 0.38
PDE4A P27815 1/20 0.38
CYP3A4 P08684 1/20 0.37
BLM P54132 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3019661 0.79 ADORA2A (0.49) ADORA1ADORA2ANQO2CYP19A1AR
SCHEMBL7978388 0.79 ADORA1 (0.61) ADORA1ADORA2ACA5ACYP3A4BLM
SCHEMBL10821728 0.76 AR (0.40) NQO2CYP19A1ARKDM4EALDH1A1
SCHEMBL11591796 0.76 ADORA1 (0.53) ADORA1ADORA2ACA5ACYP3A4BLM
SCHEMBL11590712 0.72 AR (0.55) ADORA1ADORA2AARKMT2AKDM4E
SCHEMBL29437720 0.72 AR (0.55) ADORA1ADORA2AARKMT2AKDM4E
SCHEMBL11588963 0.71 ADORA1 (0.51) ADORA1ADORA2ACA5AXDHPDE3B
SCHEMBL30681004 0.70 ADORA1 (0.47) ADORA1ADORA2ACA5AARCYP3A4
SCHEMBL1771739 0.68 AR (0.56) NQO2CYP19A1ARKDM4EALDH1A1
SCHEMBL11589180 0.67 ADORA1 (0.58) ADORA1ADORA2ACA5AXDHKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4103257-A BLUE TO NEAR ULTRAVIOLET THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 1978-07-25 US disclosed