SCHEMBL11595124

SCHEMBL11595124

COC(=O)C1CN(C2CCC(c3ccc(F)cc3)(c3ccc(F)cc3)CC2)CCC1=O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.39
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
RORC P51449 3/20 0.35
OPRL1 P41146 2/20 0.35
SLC6A3 Q01959 5/20 0.34
SLC6A2 P23975 3/20 0.34
SLC6A4 P31645 2/20 0.34
HSD11B1 P28845 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
CCR1 P32246 1/20 0.33
LIPG Q9Y5X9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL858717 0.79 BRD4 (0.36) SLC6A3SLC6A2SLC6A4
SCHEMBL551490 0.76 ALDH1A1 (0.40)
SCHEMBL11594047 0.74 CCR1 (0.41) CYP2D6RORCOPRL1HSD11B1CCR1
SCHEMBL5872111 0.68 HTR2A (0.45)
SCHEMBL5767617 0.68 PSEN1 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
Fluorobenzene SCHEMBL27495214 0.67 CHRM5 (0.51)
SCHEMBL9630718 0.67 MTNR1B (0.48)
SCHEMBL1558214 0.66 RORC (0.45) CYP2D6PSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL10395156 0.66 MTNR1B (0.47)
SCHEMBL11568317 0.66 MAPT (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4076821-A 4,4-Diphenylcycloalkylpiperidines and psychotropic compositions thereof YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JA) 1978-02-28 US disclosed