SCHEMBL11599683

SCHEMBL11599683

COc1ccc(C(=O)c2sc3ccc(OC)cc3c2-c2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.59
CNR2 P34972 5/20 0.56
CNR1 P21554 2/20 0.56
ADORA1 P30542 4/20 0.50
ALDH1A1 P00352 4/20 0.49
ADORA3 P0DMS8 3/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
HPGD P15428 1/20 0.49
CYP2C19 P33261 1/20 0.49
HTT P42858 1/20 0.49
MC4R P32245 1/20 0.48
L3MBTL1 Q9Y468 3/20 0.48
MAPT P10636 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
MAPK1 P28482 1/20 0.48
HSP90AA1 P07900 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8340562 0.90 MAOB (0.55) MAOBCNR2CNR1ADORA1ALDH1A1
SCHEMBL8335288 0.90 MAOB (0.69) MAOBCNR2CNR1ADORA1ALDH1A1
SCHEMBL11602300 0.87 L3MBTL1 (0.51) MAOBCNR2CNR1ALDH1A1CYP1A2
SCHEMBL8341825 0.86 ESR1 (0.50) MAOBCNR2CNR1ADORA1ALDH1A1
SCHEMBL11602489 0.85 EDNRA (0.49) MAOBCNR2CNR1ADORA1ALDH1A1
SCHEMBL11598733 0.83 ADORA1 (0.53) MAOBCNR2CNR1ADORA1ALDH1A1
SCHEMBL11599961 0.80 EDNRA (0.50) MAOBCNR2CNR1ALDH1A1HPGD
SCHEMBL9145308 0.80 ESR1 (0.61) MAOBMAPTMEN1KMT2ANPC1
SCHEMBL8340731 0.80 MAPT (0.49) MAOBHPGDHTTMAPTMEN1
SCHEMBL8335318 0.80 ESR1 (0.69) MAOBCNR2CNR1L3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4075227-A NONSTEROIDAL ELI LILLY AND COMPANY (US) 1978-02-21 US disclosed