SCHEMBL1160490

SCHEMBL1160490

CCNC(=O)c1ccc(N2CCN(C(C)(C)C)CC2)c(C)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.49
TNK2 Q07912 1/20 0.47
TNK1 Q13470 1/20 0.47
HTR7 P34969 1/20 0.45
DRD2 P14416 2/20 0.44
ADRA1A P35348 2/20 0.44
DRD3 P35462 2/20 0.44
NPC1 O15118 1/20 0.43
APOBEC3A P31941 1/20 0.43
RAB9A P51151 1/20 0.43
APOBEC3G Q9HC16 1/20 0.43
KMT2A Q03164 1/20 0.42
MAPK14 Q16539 2/20 0.41
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
POLB P06746 2/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1160652 0.86 PARP1 (0.46) PARP1HTR7DRD2ADRA1ADRD3
SCHEMBL2773033 0.84 PARP1 (0.50) PARP1TNK2TNK1HTR7DRD2
SCHEMBL707004 0.83 KMT2A (0.55) PARP1TNK2TNK1KMT2AHTT
SCHEMBL532364 0.82 PARP1 (0.51) PARP1TNK2TNK1HTR7NPC1
Hydrochloric Acid SCHEMBL1160638 0.81 PARP1 (0.50) PARP1TNK2TNK1HTR7NPC1
Hydrochloric Acid SCHEMBL709177 0.81 PARP1 (0.50) PARP1TNK2TNK1HTR7NPC1
SCHEMBL4151138 0.71 NR1H4 (0.61) NPC1RAB9AKMT2AMAPK14POLB
SCHEMBL16432438 0.69 IGF1R (0.43) HTR7KMT2APOLBHTTSMN1; SMN2
SCHEMBL11299409 0.69 MAPT (0.65) KMT2APOLBHTTSMN1; SMN2
SCHEMBL532249 0.69 PARP1 (0.51) PARP1TNK1DRD2DRD3HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2459561-A1 POLY (ADP-RIBOSE) POLYMERASE (PARP) INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2012-06-06 EP disclosed
WO-2011014681-A1 Poly (ADP-Ribose) Polymerase (PARP) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-02-03 WO disclosed