SCHEMBL1160652

SCHEMBL1160652

CNC(=O)c1ccc(N2CCN(C(C)(C)C)CC2)c(C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.46
SCN9A Q15858 2/20 0.43
HTR7 P34969 1/20 0.42
HTT P42858 2/20 0.41
POLB P06746 1/20 0.41
NPC1 O15118 1/20 0.41
APOBEC3A P31941 1/20 0.41
RAB9A P51151 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
HTR2A P28223 1/20 0.40
NPY2R P49146 1/20 0.40
LMNA P02545 2/20 0.39
DRD2 P14416 1/20 0.39
ADRA1A P35348 1/20 0.39
DRD3 P35462 1/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1160490 0.86 PARP1 (0.49) PARP1HTR7HTTPOLBNPC1
SCHEMBL6125348 0.83 ALDH1A3 (0.51) PARP1HTR7HTTPOLBNPC1
SCHEMBL531688 0.82 HTT (0.51) PARP1SCN9AHTR7HTTPOLB
SCHEMBL707999 0.82 LMNA (0.56) PARP1HTTPOLBLMNAALDH1A1
SCHEMBL532443 0.81 HTR3A (0.51) PARP1SCN9AHTR7HTTPOLB
Hydrochloric Acid SCHEMBL710272 0.80 HTR3A (0.50) PARP1SCN9AHTR7POLBNPC1
SCHEMBL23073596 0.75 HTR7 (0.45) PARP1SCN9AHTR7HTTPOLB
SCHEMBL11299409 0.72 MAPT (0.65) HTTPOLBLMNAALDH1A1
SCHEMBL16432438 0.72 IGF1R (0.43) HTR7HTTPOLBLMNAALDH1A1
SCHEMBL4437150 0.69 KDM4E (0.56) POLBNPC1RAB9AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2459561-A1 POLY (ADP-RIBOSE) POLYMERASE (PARP) INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2012-06-06 EP disclosed
WO-2011014681-A1 Poly (ADP-Ribose) Polymerase (PARP) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-02-03 WO disclosed