SCHEMBL11605000

SCHEMBL11605000

CSc1nc2ccnn2c2ncccc12

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.36
PDE10A Q9Y233 2/20 0.33
KMT2A Q03164 4/20 0.32
HPGD P15428 2/20 0.32
KDM4E B2RXH2 3/20 0.31
ALDH1A1 P00352 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
MEN1 O00255 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
FEN1 P39748 1/20 0.31
KDM4D Q6B0I6 2/20 0.31
TGFBR1 P36897 1/20 0.31
DYRK1A Q13627 1/20 0.31
USP2 O75604 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11608397 0.78 KMT2A (0.46) HTR6PDE10AKMT2AKDM4EALDH1A1
SCHEMBL11604789 0.76 PDE10A (0.35) PDE10AKMT2AKDM4EALDH1A1NPSR1
SCHEMBL11606253 0.76 ELANE (0.38) PDE10AKMT2AKDM4EMEN1KDM4D
SCHEMBL11603925 0.76 PDE10A (0.42) PDE10AKMT2AHPGDKDM4EALDH1A1
SCHEMBL11604755 0.76 SYK (0.36) HTR6PDE10AKMT2AKDM4EMEN1
SCHEMBL11608018 0.76 ALDH1A1 (0.34) PDE10AALDH1A1
SCHEMBL11606693 0.74 MEN1 (0.38) KMT2AHPGDMEN1L3MBTL1
SCHEMBL11602446 0.72 ACP1 (0.38) KMT2AKDM4EALDH1A1NPSR1MEN1
SCHEMBL11604780 0.71 FAAH (0.37) HPGDKDM4EALDH1A1L3MBTL1
SCHEMBL11605002 0.71 APP (0.41) KMT2AHPGDKDM4EALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4072680-A Derivatives of pyrazolo[1,5-a]pyrido[3,2-e]pyrimidine E. R. SQUIBB & SONS, INC. (US) 1978-02-07 US disclosed