SCHEMBL116126

SCHEMBL116126

COc1cc(OC)nc(NC(=O)NS(=O)(=O)Nc2ccccc2C(=O)N(C)C)n1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.55
GAA P10253 1/20 0.48
MAPT P10636 2/20 0.44
TP53 P04637 1/20 0.44
GLA P06280 1/20 0.44
CYP1A2 P05177 1/20 0.41
KMT2A Q03164 1/20 0.40
ALOX15 P16050 1/20 0.39
NAMPT P43490 1/20 0.39
HDAC1 Q13547 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29878397 1.00 CDK1 (0.55) CDK1GAAMAPTTP53GLA
Chlorobenzene SCHEMBL23797205 0.94 CDK1 (0.50) CDK1GAAMAPTTP53GLA
SCHEMBL7809237 0.94 CDK1 (0.49) CDK1GAAMAPTTP53GLA
SCHEMBL7808101 0.92 GAA (0.47) CDK1GAAMAPTTP53GLA
SCHEMBL7801275 0.90 GAA (0.45) CDK1GAAMAPTTP53GLA
SCHEMBL8380205 0.88 GAA (0.51) CDK1GAAMAPTTP53GLA
SCHEMBL8535695 0.88 GAA (0.51) CDK1GAAMAPTTP53GLA
SCHEMBL7806403 0.88 CDK1 (0.53) CDK1GAAMAPTTP53GLA
SCHEMBL7808085 0.87 GAA (0.50) CDK1GAAMAPTTP53GLA
SCHEMBL7808142 0.87 CDK1 (0.55) CDK1GAAMAPTTP53GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10837 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4713486-A1 BIOMARKERS FOR IDENTIFYING INFECTIOUS AND NON-INFECTIOUS CAUSES OF NEUROLOGICAL ILLNESS The Regents of the University of California (US) 2026-03-25 EP claimed
US-20260060254-A1 HERBICIDAL COMPOSITIONS BAYER AG (DE) 2026-03-05 US claimed
EP-4677099-A2 HERBICIDE-RESISTANT GENES FOR MITOCHONDRIAL TRANSFORMATION Napigen, Inc. (US) 2026-01-14 EP claimed
US-20260007133-A1 HERBICIDAL COMPOSITION COMPRISING AZINE COMPOUNDS BASF SE (DE) 2026-01-08 US claimed
US-12484582-B2 Herbicidal compound PRO FARM GROUP, INC. (US) 2025-12-02 US claimed
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
US-20250324976-A1 METHOD AND COMPOSITION OF SYNERGISTIC HERBICIDAL MIXTURES PRO FARM GROUP INC (US) 2025-10-23 US claimed
US-20250318528-A1 HERBICIDE COMPOSITION AND WEED CONTROLLING METHOD SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2025-10-16 US claimed
EP-4601471-A1 SUBSTITUTED 5-MEMBERED RINGS AND THEIR USE AS PESTICIDES Corteva Agriscience LLC (US) 2025-08-20 EP claimed
EP-1916889-A1 METHODS OF ALTERING POPPY CHARACTERISTICS Glaxosmithkline Australia PTY Ltd. (AU) 2008-05-07 EP claimed
WO-2007101587-A1 NEW SYNERGISTIC HERBICIDAL COMPOSITIONS ISAGRO RICERCA S.R.L. (IT) 2007-09-13 WO claimed
WO-2007079965-A2 A HERBICIDE COMPOSITION FOR PADDY FIELD BAYER CROPSCIENCE AG (DE) 2007-07-19 WO claimed
US-20070167328-A1 Herbicide Composition for Paddy Field BAYER CROPSCIENCE GMBH (DE) 2007-07-19 US claimed
WO-2007042447-A2 HERBICIDAL COMPOSITIONS BASED ON 3-PHENYLURACILS AND N-[[4-[(CYCLOPROPYLAMINO)-CARBONYL]PHENYL]SULFONYL]-2-METHOXYBENZAMIDE BASF SE (DE) 2007-04-19 WO claimed
WO-2007022561-A1 METHODS OF ALTERING POPPY CHARACTERISTICS GLAXOSMITHKLINE AUSTRALIA PTY LTD (AU) 2007-03-01 WO claimed
US-20060183638-A1 Safer control of broadleaf weeds in turf with granular formulations of ALS inhibiting herbicides CORTEVA AGRISCIENCE LLC 2006-08-17 US claimed
WO-2006086662-A2 SAFER CONTROL OF BROADLEAF WEEDS IN TURF WITH GRANULAR FORMULATIONS OF ALS INHIBITING HERBICIDES DOW AGROSCIENCES LLC (US) 2006-08-17 WO claimed
WO-2006072359-A1 SYNERGISTIC HERBICIDAL SUBSTANCE COMBINATION BAYER CROPSCIENCE AG (DE) 2006-07-13 WO claimed
EP-0971902-B1 AMINOSULFONYLUREAS WITH HERBICIDAL ACTIVITY ISAGRO RICERCA SRL (IT) 2001-12-19 EP claimed