SCHEMBL11623751

SCHEMBL11623751

CCCn1cc(C(F)(F)F)nc1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.48
DGAT1 O75907 1/20 0.45
PTGS1 P23219 3/20 0.45
TSHR P16473 1/20 0.41
NR1H3 Q13133 2/20 0.39
HSD11B1 P28845 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
NR1H2 P55055 1/20 0.39
PDE10A Q9Y233 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TLR8 Q9NR97 2/20 0.38
ADORA2A P29274 2/20 0.38
ADORA2B P29275 2/20 0.38
MAPT P10636 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA1 P30542 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1912768 0.91 TSHR (0.49) PTGS2DGAT1PTGS1TSHRNR1H3
SCHEMBL11622203 0.89 PTGS2 (0.51) PTGS2DGAT1PTGS1NR1H3HSD11B1
SCHEMBL24185707 0.85 DGAT1 (0.52) PTGS2DGAT1PTGS1NR1H3NR1H2
SCHEMBL7469586 0.80 PTGS2 (0.46) PTGS2PTGS1NR1H3RAB9ASMN1; SMN2
SCHEMBL7480252 0.79 PTGS2 (0.54) PTGS2PTGS1NR1H3HSD11B1NPC1
SCHEMBL24185637 0.77 DGAT1 (0.47) PTGS2DGAT1PTGS1TLR8ADORA2B
SCHEMBL25792141 0.74 DGAT1 (0.43) PTGS2DGAT1PTGS1NPC1RAB9A
SCHEMBL24185774 0.74 DGAT1 (0.49) PTGS2DGAT1PTGS1NR1H3NR1H2
SCHEMBL25791923 0.74 DGAT1 (0.43) PTGS2DGAT1PTGS1TLR8
SCHEMBL4882528 0.72 TLR8 (0.43) NR1H3NR1H2PDE10ATLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4125530-A FROM 1,1-DIHALO-3,3,3-TRIFLUOROACETONE, BASE, AMMONIA AND A CARBOXALDEHYDE MERCK & CO., INC. (US) 1978-11-14 US disclosed
US-4032522-A ANTI-GOUT, ANTI-HYPERURICEMIC MERCK & CO., INC. (US) 1977-06-28 US disclosed