SCHEMBL11624765

SCHEMBL11624765

O=C(OC1(c2nccc3ccccc23)CCN(Cc2ccccc2)CC1)c1ccccc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 2/20 0.81
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.46
CHRM2 P08172 4/20 0.44
CHRM3 P20309 2/20 0.44
ACHE P22303 1/20 0.43
CYP2D6 P10635 3/20 0.43
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
KDM4E B2RXH2 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
PKM P14618 1/20 0.42
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
USP2 O75604 2/20 0.41
POLB P06746 1/20 0.41
LMNA P02545 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11625232 0.85 DRD3 (0.74) DRD3MEN1KMT2APOLBNCOA3
Hydrochloric Acid SCHEMBL11623731 0.84 DRD3 (0.73) DRD3KDM4EPKMALDH1A1MEN1
SCHEMBL11625964 0.83 DRD3 (0.68) DRD3CHRM2CYP3A4TSHRCYP2C19
SCHEMBL11625386 0.83 DRD3 (0.68) DRD3ACHECYP2D6CYP3A4TSHR
SCHEMBL11627320 0.80 DRD3 (0.64) DRD3ALDH1A1LMNANCOA3
SCHEMBL11626032 0.79 OPRL1 (0.56) DRD3DRD2DRD4CHRM2ACHE
SCHEMBL6543289 0.78 OPRL1 (0.55) DRD3CHRM2CHRM3CYP2D6CYP3A4
SCHEMBL8591800 0.70 CHRM2 (0.53) DRD3DRD2DRD4CHRM2CHRM3
SCHEMBL8623218 0.70 MAPK1 (0.54) DRD3DRD2DRD4CHRM2CHRM3
SCHEMBL8623458 0.68 DRD2 (0.61) DRD3DRD2DRD4CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4122180-A Isoquinolines and anti-depressants containing them MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 1978-10-24 US disclosed