SCHEMBL11628330

SCHEMBL11628330

Nc1nc(N)c2nc(COc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)cnc2n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 12/20 1.00
FOLR1 P15328 2/20 0.72
SLC19A1 P41440 2/20 0.72
SLC46A1 Q96NT5 2/20 0.72
KDM4E B2RXH2 1/20 0.72
TLR4 O00206 1/20 0.72
MEN1 O00255 1/20 0.72
ALDH1A1 P00352 1/20 0.72
LMNA P02545 1/20 0.72
TP53 P04637 1/20 0.72
TYMS P04818 1/20 0.72
GLA P06280 1/20 0.72
POLB P06746 1/20 0.72
HMGB1 P09429 1/20 0.72
MAPT P10636 1/20 0.72
FOLR2 P14207 1/20 0.72
HPGD P15428 1/20 0.72
ALOX15 P16050 1/20 0.72
ALOX12 P18054 1/20 0.72
GART P22102 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12918463 1.00 DHFR (1.00) DHFRFOLR1SLC19A1SLC46A1KDM4E
SCHEMBL29430165 0.87 DHFR (1.00) DHFRFOLR1SLC19A1SLC46A1KDM4E
SCHEMBL15700766 0.87 DHFR (1.00) DHFRFOLR1SLC19A1SLC46A1KDM4E
SCHEMBL7081697 0.87 DHFR (1.00) DHFRFOLR1SLC19A1SLC46A1KDM4E
Aminopterin SCHEMBL29398079 0.86 DHFR (0.76) DHFRFOLR1SLC19A1SLC46A1KDM4E
Aminopterin SCHEMBL1626034 0.86 DHFR (0.76) DHFRFOLR1SLC19A1SLC46A1KDM4E
Aminopterin SCHEMBL9514067 0.86 DHFR (0.76) DHFRFOLR1SLC19A1SLC46A1KDM4E
Aminopterin SCHEMBL20769794 0.86 DHFR (0.76) DHFRFOLR1SLC19A1SLC46A1KDM4E
Aminopterin SCHEMBL29443569 0.86 DHFR (0.76) DHFRFOLR1SLC19A1SLC46A1KDM4E
Aminopterin SCHEMBL8161477 0.86 DHFR (0.76) DHFRFOLR1SLC19A1SLC46A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4079056-A REACTING 2,4-DIAMINO-6-PTERIDINE-METHANOL-HBR WITH TRIPHENYLPHOSPHINE DIBROMIDE OR PHOSPHORUS TRIBROMIDE THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH, EDUCATION AND WELFARE (US) 1978-03-14 US disclosed
US-4077957-A INTERMEDIATE FOR METHOTREXATE THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH, EDUCATION AND WELFARE (US) 1978-03-07 US disclosed