SCHEMBL11670650

SCHEMBL11670650

CCOC(=O)C1=C(N)NC(N)=C(C(=O)OC(C)C)C1c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.59
KDM4E B2RXH2 6/20 0.56
GAA P10253 2/20 0.56
PYGM P11217 2/20 0.52
PYGL P06737 1/20 0.52
CACNA1D Q01668 3/20 0.51
CACNA1F O60840 2/20 0.51
CACNA1S Q13698 2/20 0.51
CACNA1C Q13936 2/20 0.51
ALDH1A1 P00352 5/20 0.49
TSHR P16473 3/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ABCC1 P33527 1/20 0.48
KMT2A Q03164 2/20 0.47
DHFR P00374 1/20 0.47
SIRT3 Q9NTG7 1/20 0.47
HPGD P15428 2/20 0.47
LMNA P02545 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MEN1 O00255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11669396 0.92 ADORA3 (0.68) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL10684386 0.85 ADORA3 (0.75) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL14616736 0.81 ADORA3 (0.85) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL11669538 0.81 CACNA1D (0.57) ADORA3KDM4ECACNA1DCACNA1FCACNA1S
SCHEMBL11522526 0.80 CYP2C9 (0.56) ADORA3KDM4EGAAPYGMPYGL
SCHEMBL8955489 0.80 ADORA3 (0.63) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL11691621 0.80 ADORA3 (0.56) ADORA3KDM4EGAACACNA1DALDH1A1
SCHEMBL11004678 0.79 CACNA1F (0.63) ADORA3KDM4EPYGMPYGLCACNA1D
SCHEMBL3027412 0.79 ADORA3 (0.89) ADORA3KDM4EGAACACNA1DCACNA1F
SCHEMBL11688000 0.79 ADORA3 (0.62) ADORA3KDM4EGAACACNA1DCACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3957998-A ADMINISTERING BAYER AKTIENGESELLSCHAFT (DT) 1976-05-18 US claimed
US-4049662-A HYPOTENSIVE AGENTS, VASODILATORS BAYER AKTIENGESELLSCHAFT (DT) 1977-09-20 US disclosed
US-4016277-A ANTIHYPERTENSIVE AGENTS AND CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1977-04-05 US disclosed
US-4002762-A 2-Amino-3,4-dihydropyridines used to effect coronary vessel dilation and treat hypertension BAYER AKTIENGESELLSCHAFT (DT) 1977-01-11 US disclosed
US-4001252-A HYPOTENSIVES, CORONARY DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1977-01-04 US disclosed
US-3988458-A HYPOTENSIVE, CORONARY DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-10-26 US disclosed
US-3959474-A 2,6-Diamino-1,4-dihydropyridine-3,5-dicarboxylic acid esters used as coronary vessel dilators and anti-hypertensive agents BAYER AKTIENGESELLSCHAFT (DT) 1976-05-25 US disclosed
US-3957998-A ADMINISTERING BAYER AKTIENGESELLSCHAFT (DT) 1976-05-18 US disclosed
US-3950336-A HYPOTENSIVE AGENTS, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-04-13 US disclosed