SCHEMBL11680883

SCHEMBL11680883

COC(=O)CC(=O)C(=Cc1ccccc1)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.55
LMNA P02545 3/20 0.55
NPC1 O15118 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2C9 P11712 1/20 0.54
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
HTT P42858 2/20 0.50
RAB9A P51151 2/20 0.50
ALDH1A1 P00352 5/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
HPGD P15428 1/20 0.49
MAOB P27338 1/20 0.49
TP53 P04637 1/20 0.49
AGTR1 P30556 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9264709 0.86 MAPT (0.58) MAPTLMNANPC1CYP1A2CYP2C9
SCHEMBL10539201 0.78 KMT2A (0.62) MAPTNPC1MEN1KMT2AHTT
SCHEMBL28041307 0.76 GLO1 (0.62) MAPTLMNANPC1MEN1KMT2A
SCHEMBL7828363 0.74 MAPT (0.62) MAPTLMNANPC1CYP1A2CYP2C9
SCHEMBL28459461 0.74 ALDH1A1 (0.58) MAPTLMNANPC1MEN1KMT2A
SCHEMBL7828360 0.74 MAPT (0.62) MAPTLMNANPC1CYP1A2CYP2C9
SCHEMBL11216772 0.74 MAPT (0.62) MAPTLMNANPC1CYP1A2CYP2C9
Methyl Benzoate SCHEMBL29102092 0.74 MEN1 (0.71) MAPTNPC1CYP1A2MEN1KMT2A
SCHEMBL11229914 0.73 MAPT (0.50) MAPTLMNANPC1CYP1A2CYP2C9
SCHEMBL11229921 0.73 MAPT (0.50) MAPTLMNANPC1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4038399-A 1,4-DIHYDROPYRIDINE CARBOXYLIC ACID ESTERS USEFUL AS CORONARY VESSEL DILATORS AND ANTI-HYPERTENSIVES BAYER AKTIENGESELLSCHAFT (DT) 1977-07-26 US disclosed
US-4031104-A ANTIHYPERTENSIVE AGENTS BAYER AKTIENGESELLSCHAFT (DT) 1977-06-21 US disclosed
US-3996234-A CORONARY VESSEL DILATORS, HYPOTENSIVES BAYER AKTIENGESELLSCHAFT (DT) 1976-12-07 US disclosed
US-3974275-A 1,4-Dihydropyridine carboxylic acid esters useful as coronary vessel dilators and anti-hypertensives BAYER AKTIENGESELLSCHAFT (DT) 1976-08-10 US disclosed