SCHEMBL11700361

SCHEMBL11700361

NCCCCC(NSc1ccccc1[N+](=O)[O-])C(=O)O

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.69
ALDH1A1 P00352 4/20 0.69
KDM4E B2RXH2 2/20 0.69
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
GAA P10253 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
DNMT1 P26358 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43
KAT2B Q92831 2/20 0.41
LMNA P02545 2/20 0.40
ALPG P10696 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP1A2 P05177 2/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
PDE7A Q13946 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11700351 1.00 MAPT (0.69) MAPTALDH1A1KDM4EMMP2MMP9
SCHEMBL7312481 0.84 MAPT (0.78) MAPTALDH1A1KDM4EMMP2MMP9
SCHEMBL7312478 0.84 MAPT (0.78) MAPTALDH1A1KDM4EMMP2MMP9
SCHEMBL7311455 0.81 MAPT (1.00) MAPTALDH1A1KDM4EGAAMEN1
SCHEMBL7311462 0.81 MAPT (1.00) MAPTALDH1A1KDM4EGAAMEN1
SCHEMBL7540298 0.81 MAPT (0.81) MAPTALDH1A1KDM4EGAAMEN1
SCHEMBL1158293 0.80 MAPT (0.71) MAPTALDH1A1KDM4EMMP2MMP9
SCHEMBL1158294 0.80 MAPT (0.71) MAPTALDH1A1KDM4EMMP2MMP9
SCHEMBL7336052 0.79 MAPT (0.70) MAPTALDH1A1KDM4EGAAMEN1
SCHEMBL7543508 0.78 MMP2 (0.47) MAPTALDH1A1KDM4EMMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4038282-A REACTING 4-PYRIDYLCARBINOL WITH SUCCINIMIDO-CHLOROFORMATE MERCK & CO., INC. (US) 1977-07-26 US disclosed
US-4006152-A PEPTIDE INTERMEDIATE MERCK & CO., INC. (US) 1977-02-01 US disclosed
US-3950348-A INTERMEDIATE FOR PEPTIDES MERCK & CO., INC. (US) 1976-04-13 US disclosed