SCHEMBL11705358

SCHEMBL11705358

O=Cc1sccc1-c1ccc(CBr)cc1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.37
PRKDC P78527 1/20 0.32
TRPA1 O75762 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TSHR P16473 1/20 0.30
CES2 O00748 1/20 0.30
CES1 P23141 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13766280 0.83 EDNRB (0.38) PTGS1PRKDCALDH1A1
SCHEMBL6822436 0.80 PTGS1 (0.40) PTGS1PRKDCALDH1A1
SCHEMBL1829790 0.77 PTGS2 (0.45) PTGS1PRKDCALDH1A1
SCHEMBL16049525 0.77 PTGS1 (0.40) PTGS1PRKDCALDH1A1
SCHEMBL3722270 0.77 PTGS1 (0.60) PTGS1ALDH1A1
SCHEMBL2461016 0.76 BCAT2 (0.47) PTGS1PRKDCALDH1A1
SCHEMBL30940239 0.75 APP (0.41) PTGS1PRKDC
SCHEMBL9696347 0.74 PRKDC (0.41) PTGS1PRKDCALDH1A1CES1
SCHEMBL3975326 0.73 PTGS1 (0.37) PTGS1PRKDCCES1
SCHEMBL28875552 0.72 PTGS1 (0.51) PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4064132-A ANTIINFLAMMATORY AGENTS JANSSEN PHARMACEUTICA N.V. (BE) 1977-12-20 US disclosed
US-4060528-A ANTIINFLAMMATORY JANSSEN PHARMACEUTICA N.V. (BE) 1977-11-29 US disclosed
US-4035376-A ESTERS, AMIDES, HYDROXAMIC ACIDS, ANTIINFLAMMATORY JANSSEN PHARMACEUTICA N.V. (BE) 1977-07-12 US disclosed