SCHEMBL11709331

SCHEMBL11709331

COc1cccc2c1OCN(CCc1ccccc1)C2

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.50
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49
ADRA1B P35368 1/20 0.49
MAPT P10636 2/20 0.47
CYP1A2 P05177 1/20 0.46
HTR1A P08908 3/20 0.46
DRD2 P14416 1/20 0.46
SIGMAR1 Q99720 2/20 0.45
ATM Q13315 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
EBP Q15125 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL11719164 0.94 POLB (0.48) KCNH2ADRA1DADRA1AADRA1BMAPT
SCHEMBL30134682 0.90 HRH3 (0.51) KCNH2ADRA1DADRA1AADRA1BHTR1A
SCHEMBL11708757 0.90 SIGMAR1 (0.50) ADRA1DADRA1AADRA1BMAPTSIGMAR1
SCHEMBL11712922 0.90 MAPT (0.45) KCNH2ADRA1DADRA1AADRA1BMAPT
SCHEMBL11715311 0.89 DHCR7 (0.49) KCNH2ADRA1DADRA1AADRA1BMAPT
SCHEMBL11712332 0.88 CYP1A2 (0.44) KCNH2ADRA1DADRA1AADRA1BMAPT
SCHEMBL30166688 0.87 MAPT (0.43) MAPTCYP1A2HTR1ASIGMAR1GAA
SCHEMBL11708040 0.87 CYP1A2 (0.62) CYP1A2HTR1ASIGMAR1
SCHEMBL11710137 0.86 DHCR7 (0.50) ADRA1DADRA1AADRA1BMAPTSIGMAR1
SCHEMBL29362528 0.86 DHCR7 (0.50) ADRA1DADRA1AADRA1BMAPTSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4035363-A 1,3-BENZOXAZINE DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JA) 1977-07-12 US claimed
US-4035363-A 1,3-BENZOXAZINE DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JA) 1977-07-12 US disclosed