SCHEMBL11712922

SCHEMBL11712922

COc1cccc2c1OCN(CCc1ccc(C)cc1)C2

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.45
ABCB1 P08183 5/20 0.41
HRH3 Q9Y5N1 1/20 0.41
CYP3A4 P08684 1/20 0.40
KCNH2 Q12809 1/20 0.40
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
GSK3B P49841 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11708757 0.90 SIGMAR1 (0.50) MAPTABCB1HRH3ADRA1DADRA1A
SCHEMBL11709331 0.90 KCNH2 (0.50) MAPTKCNH2ADRA1DADRA1AADRA1B
SCHEMBL11715311 0.89 DHCR7 (0.49) MAPTABCB1CYP3A4KCNH2ADRA1D
SCHEMBL29362528 0.87 DHCR7 (0.50) MAPTABCB1ADRA1DADRA1AADRA1B
SCHEMBL11710137 0.87 DHCR7 (0.50) MAPTABCB1ADRA1DADRA1AADRA1B
Oxalic Acid SCHEMBL11719164 0.85 POLB (0.48) MAPTABCB1KCNH2ADRA1DADRA1A
SCHEMBL30134682 0.83 HRH3 (0.51) ABCB1HRH3KCNH2ADRA1DADRA1A
SCHEMBL30166688 0.82 MAPT (0.43) MAPTHRH3
SCHEMBL11712113 0.80 SIGMAR1 (0.43) MAPTKCNH2
SCHEMBL11707373 0.79 MAPT (0.51) MAPTABCB1HRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4035363-A 1,3-BENZOXAZINE DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JA) 1977-07-12 US claimed
US-4035363-A 1,3-BENZOXAZINE DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JA) 1977-07-12 US disclosed