SCHEMBL11710065

SCHEMBL11710065

COc1cc2c(cc1OC)C(c1ccccc1Br)NCC2

nearest known ligand 0.71

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.71
MEN1 O00255 3/20 0.71
KDM1A O60341 2/20 0.64
CA1 P00915 1/20 0.58
CA2 P00918 1/20 0.58
CA7 P43166 1/20 0.58
CA9 Q16790 1/20 0.58
CA14 Q9ULX7 1/20 0.58
ALDH1A1 P00352 2/20 0.57
LMNA P02545 1/20 0.57
MAOA P21397 2/20 0.56
TSHR P16473 1/20 0.56
DRD1 P21728 1/20 0.55
DRD5 P21918 1/20 0.55
GAA P10253 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.52
BCHE P06276 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11713664 0.84 KMT2A (0.73) KMT2AMEN1CA1CA2CA7
SCHEMBL538380 0.83 KMT2A (0.71) KMT2AMEN1CA1CA2CA7
SCHEMBL13804033 0.81 KMT2A (1.00) KMT2AMEN1KDM1ACA1CA2
SCHEMBL7849270 0.81 KMT2A (1.00) KMT2AMEN1KDM1ACA1CA2
SCHEMBL14646680 0.81 KMT2A (1.00) KMT2AMEN1KDM1ACA1CA2
SCHEMBL30789059 0.81 KMT2A (0.68) KMT2AMEN1CA1CA2CA7
SCHEMBL11714295 0.80 KMT2A (0.67) KMT2AMEN1CA1CA2CA7
Hydrochloric Acid SCHEMBL4772373 0.80 KMT2A (0.97) KMT2AMEN1KDM1ACA1CA2
SCHEMBL4024598 0.79 KMT2A (0.55) KMT2AMEN1TSHRBCHE
SCHEMBL31358960 0.78 BCHE (0.60) KMT2AMEN1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4001244-A 1-ARYL-3,4-DIHYDRO-2(1H)-ISOQUINOLINE CARBONYL CHLORIDES G. D. SEARLE & CO. (US) 1977-01-04 US disclosed