SCHEMBL11727445

SCHEMBL11727445

Cc1ccc(NC(=O)CBr)c(C(=O)c2ccccc2)c1

nearest known ligand 0.73

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.73
ALDH1A1 P00352 2/20 0.62
LMNA P02545 2/20 0.61
TP53 P04637 4/20 0.60
GAA P10253 1/20 0.60
THRB P10828 1/20 0.56
MAPK1 P28482 1/20 0.55
NPSR1 Q6W5P4 2/20 0.54
HTT P42858 2/20 0.54
MAPT P10636 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31048907 0.83 SMN1; SMN2 (0.69) ALDH1A1LMNATP53GAATHRB
SCHEMBL11538033 0.83 SMN1; SMN2 (0.69) ALDH1A1LMNATP53GAATHRB
SCHEMBL21629314 0.82 TP53 (0.73) PKMALDH1A1LMNATP53GAA
SCHEMBL29485041 0.82 ALDH1A1 (0.71) PKMALDH1A1LMNAMAPK1NPSR1
SCHEMBL8672570 0.82 ALDH1A1 (0.71) PKMALDH1A1LMNAMAPK1NPSR1
SCHEMBL19952802 0.82 PKM (0.67) PKMALDH1A1LMNATP53GAA
SCHEMBL2921293 0.81 PKM (0.64) PKMALDH1A1LMNATP53GAA
SCHEMBL28942578 0.80 ALDH1A1 (0.61) PKMALDH1A1LMNATP53GAA
SCHEMBL9379316 0.79 PKM (0.49) PKMALDH1A1LMNATP53GAA
SCHEMBL31541287 0.79 MEN1 (0.52) PKMALDH1A1LMNAGAAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4014883-A ANTITUMOR AGENTS HOFFMANN-LA ROCHE INC. (US) 1977-03-29 US disclosed