SCHEMBL11730656

SCHEMBL11730656

C1=Nc2c(ccc3ccncc23)NC1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 1/20 0.36
DYRK1A Q13627 1/20 0.36
TNF P01375 1/20 0.33
MAPK10 P53779 4/20 0.33
HIPK2 Q9H2X6 1/20 0.32
KDM4E B2RXH2 1/20 0.30
POLB P06746 1/20 0.30
HTT P42858 1/20 0.30
RAD52 P43351 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13154633 0.69 NOTUM (0.42) CLK1DYRK1ATNFMAPK10HIPK2
SCHEMBL9275580 0.69 CLK1 (0.35) CLK1DYRK1ATNFMAPK10HIPK2
SCHEMBL29569821 0.69 CLK1 (0.54) CLK1DYRK1ATNFMAPK10HIPK2
SCHEMBL672509 0.69 CLK1 (0.54) CLK1DYRK1ATNFMAPK10HIPK2
SCHEMBL8121570 0.67 GAA (0.32)
SCHEMBL12920473 0.67 CHRNB2 (0.31)
SCHEMBL8216558 0.67 CLK1 (0.39) CLK1DYRK1ATNFMAPK10HIPK2
SCHEMBL26102745 0.63 MAOA (0.37) DYRK1AHIPK2
SCHEMBL29742542 0.62 CDC7 (0.39) CLK1DYRK1ATNFMAPK10HIPK2
SCHEMBL15051861 0.62 CDC7 (0.39) CLK1DYRK1ATNFMAPK10HIPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4049659-A Process for the preparation of 4-oxo-hexahydro-pyrazinoisoquinoline derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-09-20 US claimed
US-4049659-A Process for the preparation of 4-oxo-hexahydro-pyrazinoisoquinoline derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-09-20 US disclosed