SCHEMBL11739719

SCHEMBL11739719

CC(C)COc1cccc(C(=O)CBr)c1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.55
KAT6A Q92794 2/20 0.52
FOS P01100 1/20 0.51
JUN P05412 1/20 0.51
GSK3B P49841 2/20 0.49
KMT2A Q03164 4/20 0.48
USP2 O75604 1/20 0.46
TSHR P16473 1/20 0.46
HSD17B1 P14061 1/20 0.46
HSD17B2 P37059 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.45
PTPN1 P18031 2/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
MEN1 O00255 1/20 0.45
FABP1 P07148 1/20 0.45
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16108766 0.84 NR1H4 (0.60) NR1H4KAT6AFOSJUNKMT2A
SCHEMBL1436279 0.83 NR1H4 (0.63) NR1H4KAT6AFOSJUNKMT2A
SCHEMBL931583 0.83 NR1H4 (0.75) NR1H4KAT6AFOSJUNKMT2A
SCHEMBL920107 0.83 HPGD (0.54) NR1H4KAT6AGSK3BKMT2AALDH1A1
SCHEMBL637341 0.83 KMT2A (0.54) KAT6AGSK3BKMT2APTPN1ALDH1A1
SCHEMBL7260601 0.81 PARP1 (0.60) NR1H4KAT6AFOSJUNKMT2A
SCHEMBL3248766 0.81 NR1H4 (0.58) NR1H4KAT6AFOSJUNKMT2A
SCHEMBL6705940 0.81 GSK3B (0.61) NR1H4FOSJUNGSK3BUSP2
SCHEMBL31130233 0.80 NR1H4 (0.54) NR1H4KAT6AFOSJUNKMT2A
SCHEMBL26049008 0.80 NR1H4 (0.60) NR1H4KAT6AFOSJUNKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4033978-A Thiacycl[2.2.2]azine carboxylic acids SYNTEX (U.S.A.) INC. (US) 1977-07-05 US disclosed