Bromide

Bromide

SCHEMBL1174583

Br.CN(C)CCOc1ccccc1

nearest known ligand 0.81

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 1/20 0.57
CHRM2 known ✓ P08172 1/20 0.57
ADRB1 known ✓ P08588 1/20 0.57
ADRA2A known ✓ P08913 1/20 0.57
ADRB3 known ✓ P13945 1/20 0.57
ADRA2B known ✓ P18089 1/20 0.57
CHRM3 known ✓ P20309 1/20 0.57
SLC6A2 known ✓ P23975 1/20 0.57
ADRA1D known ✓ P25100 1/20 0.57
SLC6A4 known ✓ P31645 1/20 0.57
SLC6A3 known ✓ Q01959 1/20 0.57
SIGMAR1 known ✓ Q99720 1/20 0.57
LTA4H P09960 2/20 0.81
LSS P48449 1/20 0.61
HRH3 Q9Y5N1 1/20 0.60
CHRNB2 P17787 2/20 0.59
CHRNA4 P43681 2/20 0.59
KEAP1 Q14145 1/20 0.58
NFE2L2 Q16236 1/20 0.58
KDM4E B2RXH2 3/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8494655 0.98 LTA4H (0.79) LTA4HLSSHRH3CHRNB2CHRNA4
SCHEMBL1405661 0.98 LTA4H (0.85) LTA4HLSSHRH3CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL10682691 0.96 LTA4H (0.81) LTA4HLSSHRH3CHRNB2CHRNA4
Bromide SCHEMBL8494658 0.94 LTA4H (0.79) LTA4HLSSHRH3CHRNB2CHRNA4
Ethylamine SCHEMBL9871196 0.90 LTA4H (0.73) LTA4HLSSHRH3CHRNB2CHRNA4
Tetradecane SCHEMBL28451741 0.89 LTA4H (0.67) LTA4HLSSHRH3KDM4ECYP2D6
SCHEMBL4632841 0.87 LSS (0.79) LTA4HLSSHRH3KDM4EKCNA3
Tetradecane SCHEMBL28897526 0.87 LTA4H (0.69) LTA4HLSSHRH3KDM4ECYP2D6
SCHEMBL22831331 0.86 LSS (0.83) LTA4HLSSHRH3KEAP1NFE2L2
SCHEMBL15509555 0.86 LTA4H (0.68) LTA4HLSSHRH3CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8258328-B2 Method and intermediates for preparing 19-norsteroid compounds AVENTIS PHARMA S.A. (FR) 2012-09-04 US disclosed
US-20110046402-A1 NOVEL METHOD AND INTERMEDIATES FOR PREPARING 19-NORSTEROID COMPOUNDS AVENTIS PHARMA S.A. (FR) 2011-02-24 US disclosed
US-20040229853-A1 Novel method and intermediates for preparing 19-norsteroid compounds AVENTIS PHARMA S.A. (FR) 2004-11-18 US disclosed
US-4105566-A FIREPROOFING, BIOCIDAL ACTIVITY, AMMONIUM POLYPHOSPHATE, ORGANO-TIN COMPOUND ALBRIGHT & WILSON LIMITED (GB) 1978-08-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040229853-A1 Novel method and intermediates for preparing 19-norsteroid compounds CYP17A1, HSD17B7, CYP11B1 ADRB2 267/4885CHRM2 3034/4885ADRB1 201/4885
US-20110046402-A1 NOVEL METHOD AND INTERMEDIATES FOR PREPARING 19-NORSTEROID COMPOUNDS HSD17B7, CYP17A1, HSD17B13 ADRB2 225/4885CHRM2 1624/4885ADRB1 220/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.